Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524686 (CHEMBL4470378) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.94E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50079525 (CHEMBL3417314) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50481947 (CHEBI:8416 | GNF-Pf-476 | PRISTIMERIN | Pristimeri...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 960 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50079524 (CHEMBL3417313) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524687 (CHEMBL3928971) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 830 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524688 (CHEMBL3980631) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524689 (CHEMBL4451088) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.13E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524690 (CHEMBL4463133) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.56E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50071058 ((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to purified Nur77 LBD (unknown origin) by SPR analysis | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50481949 (Dihydrocelastrol | acs.jmedchem.1c00409_ST.616) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 870 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524691 (CHEMBL4207143) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.69E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524692 (CHEMBL4470497) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524693 (CHEMBL4459092) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 720 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524694 (CHEMBL3892041) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50524695 (CHEMBL4446742) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor subfamily 4 group A member 1 (Homo sapiens (Human)) | BDBM50071058 ((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a |
Xiamen University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ... | Eur J Med Chem 177: 171-187 (2019) Article DOI: 10.1016/j.ejmech.2019.05.009 BindingDB Entry DOI: 10.7270/Q28D00P6 | |||||||||||
More data for this Ligand-Target Pair |