Compile Data Set for Download or QSAR

Found 29 hits Enz. Inhib. hit(s) with all data for entry = 50011503   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM396236 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) Show SMILES Cc1nc2nonc2c(N)c1Cc1ccc(C#N)c(NC2CC2)n1 Show InChI InChI=1S/C16H15N7O/c1-8-12(13(18)14-16(19-8)23-24-22-14)6-11-3-2-9(7-17)15(21-11)20-10-4-5-10/h2-3,10H,4-6,18H2,1H3,(H,20,21)	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0200	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548078 (CHEMBL4746798) Show SMILES Cc1nc2nonc2c(N)c1Cn1ccc(n1)-c1cccc(n1)C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0280	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548079 (CHEMBL4754865) Show SMILES COc1cc(ccc1Cc1c(C)nc2nonc2c1N)C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0660	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548076 (CHEMBL4781133 | US11583532, Example 5.1) Show SMILES Cc1nc2ncnn2c(N)c1Cc1ccc(Br)c(OC(F)F)n1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.130	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548077 (CHEMBL4789143) Show SMILES Cc1nc2nonc2c(N)c1CN1CCC(CC1)OC(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.560	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548065 (CHEMBL4785875) Show SMILES Cc1nc(ccc1COc1cc(Cl)c2cc(CC(O)=O)sc2c1Cl)C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA as substra...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548065 (CHEMBL4785875) Show SMILES Cc1nc(ccc1COc1cc(Cl)c2cc(CC(O)=O)sc2c1Cl)C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548066 (CHEMBL4791105) Show SMILES OC(=O)c1ccc2oc(SCc3ccc(Cl)cc3Cl)nc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548063 (CHEMBL4741413) Show SMILES C[C@@H](O)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CO)NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@H](CN)NC(=O)[C@H](CO)NC(=O)CN)C(N)=O |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of GOAT (unknown origin)				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548066 (CHEMBL4791105) Show SMILES OC(=O)c1ccc2oc(SCc3ccc(Cl)cc3Cl)nc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA as substra...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548069 (CHEMBL4741670) Show SMILES CCCC[C@H]1C[C@@H](C1)C(=O)NC[C@H]1CCCN1C(=O)[C@@H](NC(=S)CNC)C(C)(C)C |r,wU:12.12,6.8,wD:19.27,4.3,(17.81,-5.97,;17.5,-7.47,;18.64,-8.5,;20.11,-8.02,;21.25,-9.05,;21.33,-10.59,;22.86,-10.5,;22.79,-8.97,;24.01,-11.53,;25.48,-11.05,;23.69,-13.04,;24.84,-14.07,;24.52,-15.57,;25.55,-16.72,;24.78,-18.05,;23.28,-17.73,;23.11,-16.21,;21.77,-15.44,;21.77,-13.9,;20.44,-16.21,;19.11,-15.44,;17.77,-16.21,;17.77,-17.75,;16.44,-15.44,;15.1,-16.21,;13.77,-15.44,;20.44,-17.75,;19.11,-18.52,;21.77,-18.52,;20.42,-19.28,)| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548075 (CHEMBL4764363 | US11312709, Example 1a) Show SMILES OC(=O)Cc1csc2cc(O[C@H]3CCc4ncccc34)cc(Cl)c12 |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<50	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using biotinylated ghrelin peptide/octanoyl-CoA/palmitoyl CoA...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM367610 (N-[(1S)-2-[4-[2- (4-Amino-2- chloro-6-methyl- pyri...) Show SMILES C[C@H](NC(=O)c1cn[nH]c1C)C(=O)N1CCC(CCc2c(C)nc(Cl)nc2N)CC1 |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	54	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548061 (CHEMBL4741216) Show SMILES C[C@H](NC(=O)c1ccn(C)n1)C(=O)N1CCC(CCc2c(N)nc(N)nc2Cl)CC1 |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	69	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM289086 (N-[(1 S)-2-[4-[2-[4-Amino-6-methyl-2-(trifluoromet...) Show SMILES C[C@H](NC(=O)c1ccnn1C)C(=O)N1CCC(CCc2c(C)nc(nc2N)C(F)(F)F)CC1 |r| Show InChI InChI=1S/C21H28F3N7O2/c1-12-15(17(25)29-20(28-12)21(22,23)24)5-4-14-7-10-31(11-8-14)19(33)13(2)27-18(32)16-6-9-26-30(16)3/h6,9,13-14H,4-5,7-8,10-11H2,1-3H3,(H,27,32)(H2,25,28,29)/t13-/m0/s1	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM367612 (N-[(1S)-2-[4-[2-(4-Amino-6-chloro-2-methyl-pyrimid...) Show SMILES C[C@H](NC(=O)c1cnc(C)s1)C(=O)N1CCC(CCc2c(N)nc(C)nc2Cl)CC1 |r| Show InChI InChI=1S/C20H27ClN6O2S/c1-11(24-19(28)16-10-23-13(3)30-16)20(29)27-8-6-14(7-9-27)4-5-15-17(21)25-12(2)26-18(15)22/h10-11,14H,4-9H2,1-3H3,(H,24,28)(H2,22,25,26)/t11-/m0/s1	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	96	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM367615 (Methyl N-[(1S)-2-[4-[2-(4-amino-6-chloro-2-methyl-...) Show SMILES COC(=O)N[C@@H](C)C(=O)N1CCC(CCc2c(N)nc(C)nc2Cl)CC1 |r| Show InChI InChI=1S/C17H26ClN5O3/c1-10(20-17(25)26-3)16(24)23-8-6-12(7-9-23)4-5-13-14(18)21-11(2)22-15(13)19/h10,12H,4-9H2,1-3H3,(H,20,25)(H2,19,21,22)/t10-/m0/s1	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	149	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548062 (CHEMBL4742847) Show SMILES C[C@H](NC(=O)C1CC1)C(=O)N1CCC(CCc2c(N)nc(N)nc2Cl)CC1 |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	192	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50094876 (CHEMBL3589129) Show SMILES CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cn1cc(CCCc2ccccc2)nn1)NC(=O)[C@H](CO)NC(=O)CN)C(N)=O |r| Show InChI InChI=1S/C34H47N9O6/c1-22(2)16-26(31(36)46)38-32(47)27(17-24-12-7-4-8-13-24)39-33(48)28(40-34(49)29(21-44)37-30(45)18-35)20-43-19-25(41-42-43)15-9-14-23-10-5-3-6-11-23/h3-8,10-13,19,22,26-29,44H,9,14-18,20-21,35H2,1-2H3,(H2,36,46)(H,37,45)(H,38,47)(H,39,48)(H,40,49)/t26-,27-,28-,29-/m0/s1	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of GOAT (unknown origin) by fluorescence-based assay				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548072 (CHEMBL4778987) Show SMILES CCCCCCCC(=O)NC[C@H](NC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CN)CC(C)C |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548074 (CHEMBL4750990) Show SMILES CCCCCCCC(=O)OC[C@H](OC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCNC(N)=N)C(O)=O |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548068 (CHEMBL4753228) Show SMILES CCCCCCN(C(CNCc1ccccc1)c1ccc2cc(O)ccc2c1)C(C)=O Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM50548064 (CHEMBL4787843) Show SMILES [H][C@@]12CCC[C@@]1(C)CC[C@@]1([H])[C@@]2([H])CC[C@@]2([H])C(C)(C)C(=O)C(=C[C@]12C)C#N |r,c:24| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell membrane using GSSFLC-acrylodan and octanoyl-CoA as substrate preincubated...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Homo sapiens (Human))	BDBM217380 (CDDO-EA, 3) Show SMILES CCNC(=O)[C@]12CCC(C)(C)C[C@H]1[C@H]1C(=O)C=C3[C@@]4(C)C=C(C#N)C(=O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2 |r,t:17,21| Show InChI InChI=1S/C33H46N2O3/c1-9-35-27(38)33-14-12-28(2,3)18-21(33)25-22(36)16-24-30(6)17-20(19-34)26(37)29(4,5)23(30)10-11-31(24,7)32(25,8)13-15-33/h16-17,21,23,25H,9-15,18H2,1-8H3,(H,35,38)/t21-,23-,25-,30-,31+,32+,33-/m0/s1	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human GOAT expressed in baculovirus infected sf9 insect cell membrane using GSSFLC-acrylodan and octanoyl-CoA as substrate preincubated...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548067 (CHEMBL4762372) Show SMILES CCCCCCCCN(C(CNCc1ccccc1)c1ccc2cc(O)ccc2c1)C(C)=O Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548073 (CHEMBL4756686) Show SMILES CCCCCCCC(=O)OC[C@H](NC(=O)[C@H](CO)NC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CN)CC(C)C |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548070 (CHEMBL4784392) Show SMILES CCCCCCC[C@](C)(O)\C=C\[C@H](NC(=O)OCc1ccccc1)C(=O)OC |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Ghrelin O-acyltransferase (Mus musculus)	BDBM50548071 (CHEMBL4788110) Show SMILES CCCCCCC[C@H](O)\C=C\[C@H](NC(=O)OCc1ccccc1)C(=O)OC |r| Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human))	BDBM50548063 (CHEMBL4741413) Show SMILES C[C@@H](O)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CO)NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@H](CN)NC(=O)[C@H](CO)NC(=O)CN)C(N)=O |r| Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of GHSR-1A (unknown origin)				Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53
					More data for this Ligand-Target Pair