Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082051 (CHEMBL3422514) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082073 (CHEMBL3422407) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082065 (CHEMBL3422516) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082066 (CHEMBL3422517) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 216 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082067 (CHEMBL3422413) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082068 (CHEMBL3422414) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0800 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082069 (CHEMBL3422510) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 14 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082070 (CHEMBL3422511) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.20 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082071 (CHEMBL3422512) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 182 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082072 (CHEMBL3422513) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >500 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082075 (CHEMBL3422406) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082074 (CHEMBL3422408) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082076 (CHEMBL3422409) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082077 (CHEMBL3422410) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082078 (CHEMBL3422411) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082079 (CHEMBL3422412) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082064 (CHEMBL3422515) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair |