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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50026631   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Voltage-dependent T-type calcium channel subunit alpha-1G


(Homo sapiens (Human))		BDBM50262085
PNG
(CHEMBL468397 | methyl 5-((3-(1H-benzo[d]imidazol-2...)
Show SMILES COC(=O)C(CCCN(C)CCCc1nc2ccccc2[nH]1)(C(C)C)c1ccc(Br)cc1
Show InChI InChI=1S/C26H34BrN3O2/c1-19(2)26(25(31)32-4,20-12-14-21(27)15-13-20)16-8-18-30(3)17-7-11-24-28-22-9-5-6-10-23(22)29-24/h5-6,9-10,12-15,19H,7-8,11,16-18H2,1-4H3,(H,28,29)
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Similars
Article
PubMed
n/an/a 8.17n/an/an/an/an/an/a



Institute of Science and Technology

Curated by ChEMBL


Assay Description
Antagonist activity at T type calcium channel alpha1G (unknown origin) expressed in HEK293 cells assessed as inhibition of peak currents at 1 uM by w...

Bioorg Med Chem Lett 18: 4424-7 (2008)


Article DOI: 10.1016/j.bmcl.2008.06.037
BindingDB Entry DOI: 10.7270/Q2TT4QRD
More data for this
Ligand-Target Pair