BindingDB PrimarySearch

Found 9 hits of ph data with Target = 'Phospholipase A2, major isoenzyme'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23750 (3-{4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}-4...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23752 (3-{4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}-4,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23753 (3-{4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}-4,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23754 (3-({4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}m...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23759 (3-{4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23756 (3-({4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}me...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23757 (3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl}...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23758 (3-{4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair
Phospholipase A2, major isoenzyme (Sus scrofa (pig))	BDBM23755 (3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	22
Universite Paris 7-Denis Diderot					Assay Description PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...				Bioorg Med Chem 16: 1242-53 (2008) Article DOI: 10.1016/j.bmc.2007.10.077 BindingDB Entry DOI: 10.7270/Q2J964PK
Universite Paris 7-Denis Diderot					More data for this Ligand-Target Pair