Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154536 (2-(4-tert-butylphenyl)-1-(4-methylbenzenesulfonyl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154529 (2-(4-fluorophenyl)-1-(4-methylbenzenesulfonyl)-6-[...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154531 (2-(4-bromophenyl)-6-(4-chlorophenyl)-1-(4-methylbe...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154534 (2-(4-bromophenyl)-6-(3,4-dichlorophenyl)-1-(4-meth...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154540 (2-(4-(tert-butyl)phenyl)-N-(2-methoxyethyl)-6-(p-t...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154535 (2-(4-fluorophenyl)-1-(4-methylbenzenesulfonyl)-6-(...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154530 (1-(4-methylbenzenesulfonyl)-2-(4-methylphenyl)-6-[...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154542 (5-(bromomethyl)-6-(4-(tert-butyl)phenyl)-2-(p-toly...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.60E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154541 (N-allyl-2-(4-(tert-butyl)phenyl)-6-(p-tolyl)-1-tos...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154543 (N-((2-(4-(tert-butyl)phenyl)-6-(p-tolyl)-1-tosyl-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154533 (2-(3-chlorophenyl)-1-(4-methylbenzenesulfonyl)-6-(...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.20E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154538 (2-(4-(tert-butyl)phenyl)-N-cyclopropyl-6-(p-tolyl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.30E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154532 (2-(3-chlorophenyl)-6-(4-ethylphenyl)-1-(4-methylbe...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154539 (2-(4-(tert-butyl)phenyl)-N-cyclohexyl-6-(p-tolyl)-...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154537 (2-(4-(tert-butyl)phenyl)-N-methyl-6-(p-tolyl)-1-to...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor acetylhydrolase IB subunit alpha2 (Mus musculus (Mouse)) | BDBM154544 (Methyl-2-(4-(tert-butyl)phenyl)-6-(p-tolyl)-1-tosy...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | n/a |
University of California, Berkeley | Assay Description For in vitro experiments, proteomes were diluted to 1 mg/mL in PBS (pH 7.5, 50 μL total reaction volume), doped with 1 μM recombinant PAFAH... | ACS Chem Biol 10: 925-32 (2015) Article DOI: 10.1021/cb500893q BindingDB Entry DOI: 10.7270/Q2CJ8C6T | |||||||||||
More data for this Ligand-Target Pair |