Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107307 (US8592379, 19) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107314 (US8592379, 36 | US8592379, 37) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107306 (US8592379, 1) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107308 (US8592379, 20) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107309 (US8592379, 21) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107312 (US8592379, 24a/24b | US8592379, 35) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107310 (US8592379, 22 | US8592379, 33) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107314 (US8592379, 36 | US8592379, 37) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107312 (US8592379, 24a/24b | US8592379, 35) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM47092 (US8592379, 23) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
KiSS-1 receptor (Homo sapiens (Human)) | BDBM107316 (US8592379, 26) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University; Takeda Pharmaceutical Company Limited US Patent | Assay Description Binding inhibition assay using human GPR54. | US Patent US8592379 (2013) BindingDB Entry DOI: 10.7270/Q2N0156N | |||||||||||
More data for this Ligand-Target Pair |