Affinity Data by PubMed id=10633034

PubMed code 10633034

Found 5 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50354849 (CCI-18781 \| Cutivate \| FLUTICASONE PROPIONATE \| Fl...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE PC cid PC sid UniChem Patents Similars	DrugBank PubMed	n/a	n/a	0.5	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Research and Development Curated by ChEMBL					Assay Description Inhibition of [3H]-dexamethasone binding to human Glucocorticoid Receptor				J Med Chem 43: 19-21 (2000) BindingDB Entry DOI: 10.7270/Q2DR2TPK
Glaxo Wellcome Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50083757 (CHEMBL302366 \| Isomer of 4b,12-Difluoro-5-hydroxy-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Research and Development Curated by ChEMBL					Assay Description Inhibition of [3H]-dexamethasone binding to human Glucocorticoid Receptor				J Med Chem 43: 19-21 (2000) BindingDB Entry DOI: 10.7270/Q2DR2TPK
Glaxo Wellcome Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50083757 (CHEMBL302366 \| Isomer of 4b,12-Difluoro-5-hydroxy-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Research and Development Curated by ChEMBL					Assay Description Inhibition of [3H]-dexamethasone binding to human Glucocorticoid Receptor				J Med Chem 43: 19-21 (2000) BindingDB Entry DOI: 10.7270/Q2DR2TPK
Glaxo Wellcome Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50083758 (CHEMBL63241 \| Sodium Salt of 2-[2-(4b,12-Difluoro-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	194	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Research and Development Curated by ChEMBL					Assay Description Inhibition of [3H]-dexamethasone binding to human Glucocorticoid Receptor				J Med Chem 43: 19-21 (2000) BindingDB Entry DOI: 10.7270/Q2DR2TPK
Glaxo Wellcome Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50083758 (CHEMBL63241 \| Sodium Salt of 2-[2-(4b,12-Difluoro-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	827	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Research and Development Curated by ChEMBL					Assay Description Inhibition of [3H]-dexamethasone binding to human Glucocorticoid Receptor				J Med Chem 43: 19-21 (2000) BindingDB Entry DOI: 10.7270/Q2DR2TPK
Glaxo Wellcome Research and Development Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%