Affinity Data by PubMed id=19447628

PubMed code 19447628

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298243 ((2E,6E)-8-(2-diazo-3,3,3-trifluoropropanoyloxy)-3,...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem	Article PubMed	200	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298245 (4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	480	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298242 ((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	610	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298243 ((2E,6E)-8-(2-diazo-3,3,3-trifluoropropanoyloxy)-3,...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	720	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298245 (4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298242 ((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha (Saccharomyces cerevisiae)	BDBM50298244 (3-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Minnesota Curated by ChEMBL					Assay Description Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIA				Bioorg Med Chem 17: 4797-805 (2009) Article DOI: 10.1016/j.bmc.2009.04.034 BindingDB Entry DOI: 10.7270/Q2HT2PCH
University of Minnesota Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%