Found 20 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353649
(CHEMBL1829835)Show SMILES OC(=O)CC(Cc1nc2ccc(I)cc2[nH]1)c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C17H13Cl2IN2O2/c18-12-3-1-9(5-13(12)19)10(7-17(23)24)6-16-21-14-4-2-11(20)8-15(14)22-16/h1-5,8,10H,6-7H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353651
(CHEMBL1829841)Show SMILES CC(C)(C)c1ccc(cc1)C(CC(O)=O)Cc1nc2ccc(I)cc2[nH]1 Show InChI InChI=1S/C21H23IN2O2/c1-21(2,3)15-6-4-13(5-7-15)14(11-20(25)26)10-19-23-17-9-8-16(22)12-18(17)24-19/h4-9,12,14H,10-11H2,1-3H3,(H,23,24)(H,25,26) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353652
(CHEMBL1829842)Show SMILES CCCc1ccc(cc1)C(CC(O)=O)Cc1nc2ccc(I)cc2[nH]1 Show InChI InChI=1S/C20H21IN2O2/c1-2-3-13-4-6-14(7-5-13)15(11-20(24)25)10-19-22-17-9-8-16(21)12-18(17)23-19/h4-9,12,15H,2-3,10-11H2,1H3,(H,22,23)(H,24,25) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353647
(CHEMBL1829832)Show SMILES OC(=O)CC(Cc1nc2cc(Cl)cc(Cl)c2[nH]1)c1ccc(Cl)cc1 Show InChI InChI=1S/C17H13Cl3N2O2/c18-11-3-1-9(2-4-11)10(6-16(23)24)5-15-21-14-8-12(19)7-13(20)17(14)22-15/h1-4,7-8,10H,5-6H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
PDB
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353653
(CHEMBL1829843)Show SMILES OC(=O)CC(Cc1nc2ccc(cc2[nH]1)-c1ccccc1)c1ccc(Cl)cc1 Show InChI InChI=1S/C23H19ClN2O2/c24-19-9-6-16(7-10-19)18(14-23(27)28)13-22-25-20-11-8-17(12-21(20)26-22)15-4-2-1-3-5-15/h1-12,18H,13-14H2,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353649
(CHEMBL1829835)Show SMILES OC(=O)CC(Cc1nc2ccc(I)cc2[nH]1)c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C17H13Cl2IN2O2/c18-12-3-1-9(5-13(12)19)10(7-17(23)24)6-16-21-14-4-2-11(20)8-15(14)22-16/h1-5,8,10H,6-7H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353653
(CHEMBL1829843)Show SMILES OC(=O)CC(Cc1nc2ccc(cc2[nH]1)-c1ccccc1)c1ccc(Cl)cc1 Show InChI InChI=1S/C23H19ClN2O2/c24-19-9-6-16(7-10-19)18(14-23(27)28)13-22-25-20-11-8-17(12-21(20)26-22)15-4-2-1-3-5-15/h1-12,18H,13-14H2,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353651
(CHEMBL1829841)Show SMILES CC(C)(C)c1ccc(cc1)C(CC(O)=O)Cc1nc2ccc(I)cc2[nH]1 Show InChI InChI=1S/C21H23IN2O2/c1-21(2,3)15-6-4-13(5-7-15)14(11-20(25)26)10-19-23-17-9-8-16(22)12-18(17)24-19/h4-9,12,14H,10-11H2,1-3H3,(H,23,24)(H,25,26) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353653
(CHEMBL1829843)Show SMILES OC(=O)CC(Cc1nc2ccc(cc2[nH]1)-c1ccccc1)c1ccc(Cl)cc1 Show InChI InChI=1S/C23H19ClN2O2/c24-19-9-6-16(7-10-19)18(14-23(27)28)13-22-25-20-11-8-17(12-21(20)26-22)15-4-2-1-3-5-15/h1-12,18H,13-14H2,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353653
(CHEMBL1829843)Show SMILES OC(=O)CC(Cc1nc2ccc(cc2[nH]1)-c1ccccc1)c1ccc(Cl)cc1 Show InChI InChI=1S/C23H19ClN2O2/c24-19-9-6-16(7-10-19)18(14-23(27)28)13-22-25-20-11-8-17(12-21(20)26-22)15-4-2-1-3-5-15/h1-12,18H,13-14H2,(H,25,26)(H,27,28) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353650
(CHEMBL1829837)Show SMILES OC(=O)CC(Cc1nc2ccc(Cl)cc2[nH]1)c1ccc(Cl)c(c1)C(F)(F)F Show InChI InChI=1S/C18H13Cl2F3N2O2/c19-11-2-4-14-15(8-11)25-16(24-14)6-10(7-17(26)27)9-1-3-13(20)12(5-9)18(21,22)23/h1-5,8,10H,6-7H2,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353648
(CHEMBL1829833)Show SMILES Cc1cc(Cl)cc2[nH]c(CC(CC(O)=O)c3ccc(Cl)cc3)nc12 Show InChI InChI=1S/C18H16Cl2N2O2/c1-10-6-14(20)9-15-18(10)22-16(21-15)7-12(8-17(23)24)11-2-4-13(19)5-3-11/h2-6,9,12H,7-8H2,1H3,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353655
(CHEMBL1829834)Show SMILES OC(=O)CC(Cc1nc2ccc(Cl)cc2[nH]1)c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C17H13Cl3N2O2/c18-11-2-4-14-15(8-11)22-16(21-14)6-10(7-17(23)24)9-1-3-12(19)13(20)5-9/h1-5,8,10H,6-7H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353654
(CHEMBL1829822)Show InChI InChI=1S/C17H14ClIN2O2/c18-12-3-1-10(2-4-12)11(8-17(22)23)7-16-20-14-6-5-13(19)9-15(14)21-16/h1-6,9,11H,7-8H2,(H,20,21)(H,22,23) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353652
(CHEMBL1829842)Show SMILES CCCc1ccc(cc1)C(CC(O)=O)Cc1nc2ccc(I)cc2[nH]1 Show InChI InChI=1S/C20H21IN2O2/c1-2-3-13-4-6-14(7-5-13)15(11-20(24)25)10-19-22-17-9-8-16(21)12-18(17)23-19/h4-9,12,15H,2-3,10-11H2,1H3,(H,22,23)(H,24,25) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353647
(CHEMBL1829832)Show SMILES OC(=O)CC(Cc1nc2cc(Cl)cc(Cl)c2[nH]1)c1ccc(Cl)cc1 Show InChI InChI=1S/C17H13Cl3N2O2/c18-11-3-1-9(2-4-11)10(6-16(23)24)5-15-21-14-8-12(19)7-13(20)17(14)22-15/h1-4,7-8,10H,5-6H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
PDB
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353654
(CHEMBL1829822)Show InChI InChI=1S/C17H14ClIN2O2/c18-12-3-1-10(2-4-12)11(8-17(22)23)7-16-20-14-6-5-13(19)9-15(14)21-16/h1-6,9,11H,7-8H2,(H,20,21)(H,22,23) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assay |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353655
(CHEMBL1829834)Show SMILES OC(=O)CC(Cc1nc2ccc(Cl)cc2[nH]1)c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C17H13Cl3N2O2/c18-11-2-4-14-15(8-11)22-16(21-14)6-10(7-17(23)24)9-1-3-12(19)13(20)5-9/h1-5,8,10H,6-7H2,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353650
(CHEMBL1829837)Show SMILES OC(=O)CC(Cc1nc2ccc(Cl)cc2[nH]1)c1ccc(Cl)c(c1)C(F)(F)F Show InChI InChI=1S/C18H13Cl2F3N2O2/c19-11-2-4-14-15(8-11)25-16(24-14)6-10(7-17(26)27)9-1-3-13(20)12(5-9)18(21,22)23/h1-5,8,10H,6-7H2,(H,24,25)(H,26,27) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 4.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
Protein kinase C zeta type
(Homo sapiens (Human)) | BDBM50353648
(CHEMBL1829833)Show SMILES Cc1cc(Cl)cc2[nH]c(CC(CC(O)=O)c3ccc(Cl)cc3)nc12 Show InChI InChI=1S/C18H16Cl2N2O2/c1-10-6-14(20)9-15-18(10)22-16(21-15)7-12(8-17(23)24)11-2-4-13(19)5-3-11/h2-6,9,12H,7-8H2,1H3,(H,21,22)(H,23,24) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University
Curated by ChEMBL
| Assay Description
Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrate |
J Med Chem 54: 6714-23 (2011)
Article DOI: 10.1021/jm2005892
BindingDB Entry DOI: 10.7270/Q2CJ8DVR |
More data for this
Ligand-Target Pair | |
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