Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ras-related C3 botulinum toxin substrate 1 (Homo sapiens (Human)) | BDBM50007190 (CHEMBL3237589) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of Rac1 in human MDA-MB-435 cells after 24 hrs by G-LISA assay | J Med Chem 57: 2953-62 (2014) Article DOI: 10.1021/jm401924s BindingDB Entry DOI: 10.7270/Q2D2204K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Homo sapiens (Human)) | BDBM50007189 (CHEMBL3237582) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of Rac1 in human MDA-MB-435 cells after 24 hrs by G-LISA assay | J Med Chem 57: 2953-62 (2014) Article DOI: 10.1021/jm401924s BindingDB Entry DOI: 10.7270/Q2D2204K | |||||||||||
More data for this Ligand-Target Pair |