Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012133 (CHEMBL3263699) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012129 (CHEMBL3264012) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012125 (CHEMBL3263715) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012134 (CHEMBL3263700) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H]T0901317 from LXRbeta (unknown origin) | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012135 (CHEMBL3263701) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012142 (CHEMBL3263711) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012132 (CHEMBL3263698) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 920 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012127 (CHEMBL3263717) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012131 (CHEMBL3263697) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012143 (CHEMBL3263712) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012138 (CHEMBL3263704) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012128 (CHEMBL3264011) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012139 (CHEMBL3263707) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012137 (CHEMBL3263703) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012136 (CHEMBL3263702) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012144 (CHEMBL3263713) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012146 (CHEMBL3263706) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012145 (CHEMBL3263705) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012140 (CHEMBL3263708) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012141 (CHEMBL3263709) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation counting | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Displacement of [3H]T0901317 from LXRalpha (unknown origin) | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 450 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORa expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012131 (CHEMBL3263697) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012143 (CHEMBL3263712) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012127 (CHEMBL3263717) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORa expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity a... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012137 (CHEMBL3263703) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012144 (CHEMBL3263713) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORa expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012136 (CHEMBL3263702) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012140 (CHEMBL3263708) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 470 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORa expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity a... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012124 (CHEMBL3263714) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity a... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012125 (CHEMBL3263715) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 460 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012132 (CHEMBL3263698) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012134 (CHEMBL3263700) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012135 (CHEMBL3263701) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012141 (CHEMBL3263709) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 360 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012139 (CHEMBL3263707) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012142 (CHEMBL3263711) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 360 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012128 (CHEMBL3264011) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012129 (CHEMBL3264012) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012138 (CHEMBL3263704) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012133 (CHEMBL3263699) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity a... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM50012123 (CHEMBL3263696) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity a... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-beta (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012130 (CHEMBL3263710) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 21 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3... | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50012126 (CHEMBL3263716) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-alpha (Homo sapiens (Human)) | BDBM50012122 (CHEMBL3263695) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Inverse agonist activity at human GAL4-fused RORa expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assay | Bioorg Med Chem Lett 24: 2182-7 (2014) Article DOI: 10.1016/j.bmcl.2014.03.038 BindingDB Entry DOI: 10.7270/Q29K4CSN | |||||||||||
More data for this Ligand-Target Pair |