Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284800 (((5R,6S)-9-Bromo-6-ethyl-2,3-dioxo-2,3,6,7-tetrahy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50038046 (2-((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284808 (2-((5R,6S)-9-Bromo-6-methyl-2,3-dioxo-2,3,6,7-tetr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284801 (((5R,6S)-9-Bromo-6-methyl-2,3-dioxo-2,3,6,7-tetrah...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284805 (2-((5R,6S)-9-Bromo-6-ethyl-2,3-dioxo-2,3,6,7-tetra...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284804 (2-((5S,7R)-9-Bromo-7-methyl-2,3-dioxo-2,3,6,7-tetr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284807 (((5R,6R)-9-Bromo-6-isopropyl-2,3-dioxo-2,3,6,7-tet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50038055 (((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-py...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 9.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284806 (2-((5S,7S)-9-Bromo-7-methyl-2,3-dioxo-2,3,6,7-tetr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284799 (2-((5R,6R)-9-Bromo-6-methyl-2,3-dioxo-2,3,6,7-tetr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284798 (((5R,6R)-9-Bromo-6-methyl-2,3-dioxo-2,3,6,7-tetrah...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284812 (((5S,7R)-9-Bromo-7-methyl-2,3-dioxo-2,3,6,7-tetrah...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284811 (((5S,7S)-9-Bromo-7-methyl-2,3-dioxo-2,3,6,7-tetrah...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284803 (2-((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 241 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284803 (2-((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 241 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284810 (((S)-9-Bromo-5-methyl-2,3-dioxo-2,3,6,7-tetrahydro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 451 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284802 (2-((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 665 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284802 (2-((S)-9-Bromo-2,3-dioxo-2,3,6,7-tetrahydro-1H,5H-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 665 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50284809 (2-((S)-9-Bromo-5-methyl-2,3-dioxo-2,3,6,7-tetrahyd...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | 760 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Affinity measured by using [3H]5,7-dichlorokynurenic acid (DCKA) for the glycine binding site of NMDA receptor | Bioorg Med Chem Lett 5: 1527-1532 (1995) Article DOI: 10.1016/0960-894X(95)00243-M BindingDB Entry DOI: 10.7270/Q2K35TKC | |||||||||||
More data for this Ligand-Target Pair |