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USPatent US8629158

Compile data set for download or QSAR
Found 46 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112722
PNG
(US8629158, 36)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C25H21F3N4O/c1-31-20-12-17(4-5-18(20)24-19-6-3-16(30-19)11-21(24)31)32-9-8-14(10-23(32)33)15-2-7-22(29-13-15)25(26,27)28/h2,4-5,7-10,12-13,16,19,30H,3,6,11H2,1H3
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US Patent
 5.30 -47.2n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112692
PNG
(US8629158, 5)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(nc1)C(F)(F)F |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H21F3N4O/c1-31-20-12-17(4-5-18(20)24-19-6-3-16(30-19)11-21(24)31)32-9-8-14(10-23(32)33)15-2-7-22(29-13-15)25(26,27)28/h2,4-5,7-10,12-13,16,19,30H,3,6,11H2,1H3
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US Patent
 6.5 -46.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112693
PNG
(US8629158, 24 | US8629158, 25 | US8629158, 6)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(F)cn2)cc1=O |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H23FN4O2/c1-29-22-11-18(5-6-20(22)25-21-7-4-16(28-21)10-23(25)29)30-9-8-19(12-24(30)31)32-14-17-3-2-15(26)13-27-17/h2-3,5-6,8-9,11-13,16,21,28H,4,7,10,14H2,1H3
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US Patent
 7.40 -46.4n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112701
PNG
(US8629158, 14 | US8629158, 15)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C26H25N3O2/c1-28-23-14-19(8-9-21(23)26-22-10-7-18(27-22)13-24(26)28)29-12-11-20(15-25(29)30)31-16-17-5-3-2-4-6-17/h2-6,8-9,11-12,14-15,18,22,27H,7,10,13,16H2,1H3
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US Patent
 7.80 -46.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112695
PNG
(US8629158, 20 | US8629158, 21 | US8629158, 8)
Show SMILES O=c1cc(OCc2ccccc2)ccn1-c1ccc2c3C4CCC(Cc3[nH]c2c1)N4
Show InChI InChI=1S/C25H23N3O2/c29-24-14-19(30-15-16-4-2-1-3-5-16)10-11-28(24)18-7-8-20-22(13-18)27-23-12-17-6-9-21(26-17)25(20)23/h1-5,7-8,10-11,13-14,17,21,26-27H,6,9,12,15H2
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 9.30 -45.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112699
PNG
(US8629158, 12)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C27H27N3O2/c1-29-24-15-20(10-11-22(24)27-23-9-5-8-19(28-23)14-25(27)29)30-13-12-21(16-26(30)31)32-17-18-6-3-2-4-7-18/h2-4,6-7,10-13,15-16,19,23,28H,5,8-9,14,17H2,1H3
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 9.30 -45.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112713
PNG
(US8629158, 26)
Show SMILES CN1C2CCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C27H27N3O2/c1-28-19-9-11-23(28)27-22-10-8-20(15-24(22)29(2)25(27)14-19)30-13-12-21(16-26(30)31)32-17-18-6-4-3-5-7-18/h3-8,10,12-13,15-16,19,23H,9,11,14,17H2,1-2H3
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 9.70 -45.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112695
PNG
(US8629158, 20 | US8629158, 21 | US8629158, 8)
Show SMILES O=c1cc(OCc2ccccc2)ccn1-c1ccc2c3C4CCC(Cc3[nH]c2c1)N4
Show InChI InChI=1S/C25H23N3O2/c29-24-14-19(30-15-16-4-2-1-3-5-16)10-11-28(24)18-7-8-20-22(13-18)27-23-12-17-6-9-21(26-17)25(20)23/h1-5,7-8,10-11,13-14,17,21,26-27H,6,9,12,15H2
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US Patent
 9.80 -45.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112689
PNG
(US8629158, 2)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccccc2)cc1=O |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C26H25N3O2/c1-28-23-14-19(8-9-21(23)26-22-10-7-18(27-22)13-24(26)28)29-12-11-20(15-25(29)30)31-16-17-5-3-2-4-6-17/h2-6,8-9,11-12,14-15,18,22,27H,7,10,13,16H2,1H3
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 10.5 -45.5n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112715
PNG
(US8629158, 28)
Show SMILES CC(C)N1C2CCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C29H31N3O2/c1-19(2)32-22-10-12-25(32)29-24-11-9-21(15-26(24)30(3)27(29)16-22)31-14-13-23(17-28(31)33)34-18-20-7-5-4-6-8-20/h4-9,11,13-15,17,19,22,25H,10,12,16,18H2,1-3H3
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 12 -45.2n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112723
PNG
(US8629158, 38)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(nc2)C(F)(F)F)cc1=O
Show InChI InChI=1S/C26H23F3N4O2/c1-32-21-11-17(4-5-19(21)25-20-6-3-16(31-20)10-22(25)32)33-9-8-18(12-24(33)34)35-14-15-2-7-23(30-13-15)26(27,28)29/h2,4-5,7-9,11-13,16,20,31H,3,6,10,14H2,1H3
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 12 -45.2n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112706
PNG
(US8629158, 19)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(nc2)C(F)(F)F)cc1=O
Show InChI InChI=1S/C27H25F3N4O2/c1-33-22-12-18(6-7-20(22)26-21-4-2-3-17(32-21)11-23(26)33)34-10-9-19(13-25(34)35)36-15-16-5-8-24(31-14-16)27(28,29)30/h5-10,12-14,17,21,32H,2-4,11,15H2,1H3
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 13 -45.0n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112693
PNG
(US8629158, 24 | US8629158, 25 | US8629158, 6)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(F)cn2)cc1=O |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H23FN4O2/c1-29-22-11-18(5-6-20(22)25-21-7-4-16(28-21)10-23(25)29)30-9-8-19(12-24(30)31)32-14-17-3-2-15(26)13-27-17/h2-3,5-6,8-9,11-13,16,21,28H,4,7,10,14H2,1H3
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 13.5 -44.9n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112718
PNG
(US8629158, 31)
Show SMILES CN1C2CCCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C28H29N3O2/c1-29-20-9-6-10-24(29)28-23-12-11-21(16-25(23)30(2)26(28)15-20)31-14-13-22(17-27(31)32)33-18-19-7-4-3-5-8-19/h3-5,7-8,11-14,16-17,20,24H,6,9-10,15,18H2,1-2H3
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 14 -44.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112732
PNG
(US8629158, 47)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccc(Cl)cc2F)cc1=O
Show InChI InChI=1S/C25H22ClFN4O2/c1-30-21-11-16-4-6-20(28-16)24(21)18-5-7-22(29-25(18)30)31-9-8-17(12-23(31)32)33-13-14-2-3-15(26)10-19(14)27/h2-3,5,7-10,12,16,20,28H,4,6,11,13H2,1H3
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 14 -44.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112691
PNG
(US8629158, 16 | US8629158, 4)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(cn1)C(F)(F)F |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H21F3N4O/c1-31-21-12-17(4-5-18(21)24-20-7-3-16(30-20)11-22(24)31)32-9-8-14(10-23(32)33)19-6-2-15(13-29-19)25(26,27)28/h2,4-6,8-10,12-13,16,20,30H,3,7,11H2,1H3
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 14 -44.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112719
PNG
(US8629158, 32)
Show SMILES CCN1C2CCCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C29H31N3O2/c1-3-31-21-10-7-11-25(31)29-24-13-12-22(16-26(24)30(2)27(29)17-21)32-15-14-23(18-28(32)33)34-19-20-8-5-4-6-9-20/h4-6,8-9,12-16,18,21,25H,3,7,10-11,17,19H2,1-2H3
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 15 -44.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112701
PNG
(US8629158, 14 | US8629158, 15)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C26H25N3O2/c1-28-23-14-19(8-9-21(23)26-22-10-7-18(27-22)13-24(26)28)29-12-11-20(15-25(29)30)31-16-17-5-3-2-4-6-17/h2-6,8-9,11-12,14-15,18,22,27H,7,10,13,16H2,1H3
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 15.8 -44.5n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112691
PNG
(US8629158, 16 | US8629158, 4)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(cn1)C(F)(F)F |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H21F3N4O/c1-31-21-12-17(4-5-18(21)24-20-7-3-16(30-20)11-22(24)31)32-9-8-14(10-23(32)33)19-6-2-15(13-29-19)25(26,27)28/h2,4-6,8-10,12-13,16,20,30H,3,7,11H2,1H3
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 16.1 -44.5n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112710
PNG
(US8629158, 23)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccccn2)cc1=O
Show InChI InChI=1S/C25H24N4O2/c1-28-22-13-18(6-7-20(22)25-21-8-5-16(27-21)12-23(25)28)29-11-9-19(14-24(29)30)31-15-17-4-2-3-10-26-17/h2-4,6-7,9-11,13-14,16,21,27H,5,8,12,15H2,1H3
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 17 -44.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112720
PNG
(US8629158, 33)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)N1CCN(CCc2ccccc2)CC1=O
Show InChI InChI=1S/C26H30N4O/c1-28-23-16-20(8-9-21(23)26-22-10-7-19(27-22)15-24(26)28)30-14-13-29(17-25(30)31)12-11-18-5-3-2-4-6-18/h2-6,8-9,16,19,22,27H,7,10-15,17H2,1H3
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 17 -44.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112734
PNG
(US8629158, 50)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(cc1=O)-c1ccc(cc1)C(F)(F)F
Show InChI InChI=1S/C25H21F3N4O/c1-31-20-13-17-6-8-19(29-17)23(20)18-7-9-21(30-24(18)31)32-11-10-15(12-22(32)33)14-2-4-16(5-3-14)25(26,27)28/h2-5,7,9-12,17,19,29H,6,8,13H2,1H3
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 19 -44.1n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112693
PNG
(US8629158, 24 | US8629158, 25 | US8629158, 6)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(F)cn2)cc1=O |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H23FN4O2/c1-29-22-11-18(5-6-20(22)25-21-7-4-16(28-21)10-23(25)29)30-9-8-19(12-24(30)31)32-14-17-3-2-15(26)13-27-17/h2-3,5-6,8-9,11-13,16,21,28H,4,7,10,14H2,1H3
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 19 -44.1n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112724
PNG
(US8629158, 39)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccccc2)cc1=O |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C25H24N4O2/c1-28-21-13-17-7-9-20(26-17)24(21)19-8-10-22(27-25(19)28)29-12-11-18(14-23(29)30)31-15-16-5-3-2-4-6-16/h2-6,8,10-12,14,17,20,26H,7,9,13,15H2,1H3
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 21 -43.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112698
PNG
(US8629158, 11)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(cc12)-n1ccc(OCc2ccc(F)cn2)cc1=O
Show InChI InChI=1S/C26H25FN4O2/c1-30-23-12-19(7-8-21(23)26-22-4-2-3-17(29-22)11-24(26)30)31-10-9-20(13-25(31)32)33-15-18-6-5-16(27)14-28-18/h5-10,12-14,17,22,29H,2-4,11,15H2,1H3
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 21.3 -43.8n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112697
PNG
(US8629158, 10)
Show SMILES FC(F)(F)c1ccc(cn1)-c1ccn(-c2ccc3c4C5CCC(Cc4[nH]c3c2)N5)c(=O)c1 |THB:17:18:28:20.21,25:24:28:20.21|
Show InChI InChI=1S/C24H19F3N4O/c25-24(26,27)21-6-1-14(12-28-21)13-7-8-31(22(32)9-13)16-3-4-17-19(11-16)30-20-10-15-2-5-18(29-15)23(17)20/h1,3-4,6-9,11-12,15,18,29-30H,2,5,10H2
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 22.7 -43.6n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112690
PNG
(US8629158, 3)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(nn1)C(F)(F)F |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C24H20F3N5O/c1-31-19-12-15(3-4-16(19)23-18-5-2-14(28-18)11-20(23)31)32-9-8-13(10-22(32)33)17-6-7-21(30-29-17)24(25,26)27/h3-4,6-10,12,14,18,28H,2,5,11H2,1H3
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 24.4 -43.5n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112709
PNG
(US8629158, 22)
Show SMILES O=c1cc(OCc2ccccn2)ccn1-c1ccc2c3C4CCC(Cc3[nH]c2c1)N4
Show InChI InChI=1S/C24H22N4O2/c29-23-13-18(30-14-16-3-1-2-9-25-16)8-10-28(23)17-5-6-19-21(12-17)27-22-11-15-4-7-20(26-15)24(19)22/h1-3,5-6,8-10,12-13,15,20,26-27H,4,7,11,14H2
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 25 -43.4n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112696
PNG
(US8629158, 9)
Show SMILES Fc1ccc(COc2ccn(-c3ccc4c5C6CCC(Cc5[nH]c4c3)N6)c(=O)c2)nc1
Show InChI InChI=1S/C24H21FN4O2/c25-14-1-2-16(26-12-14)13-31-18-7-8-29(23(30)11-18)17-4-5-19-21(10-17)28-22-9-15-3-6-20(27-15)24(19)22/h1-2,4-5,7-8,10-12,15,20,27-28H,3,6,9,13H2
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 25.3 -43.4n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112730
PNG
(US8629158, 45)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccc(F)cc2F)cc1=O
Show InChI InChI=1S/C25H22F2N4O2/c1-30-21-11-16-4-6-20(28-16)24(21)18-5-7-22(29-25(18)30)31-9-8-17(12-23(31)32)33-13-14-2-3-15(26)10-19(14)27/h2-3,5,7-10,12,16,20,28H,4,6,11,13H2,1H3
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 26 -43.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112727
PNG
(US8629158, 42)
Show SMILES CN1C2CCC1c1c(C2)n(C)c2nc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C26H26N4O2/c1-28-18-8-10-21(28)25-20-9-11-23(27-26(20)29(2)22(25)14-18)30-13-12-19(15-24(30)31)32-16-17-6-4-3-5-7-17/h3-7,9,11-13,15,18,21H,8,10,14,16H2,1-2H3
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 27 -43.2n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112733
PNG
(US8629158, 48)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccc(Cl)cc2Cl)cc1=O
Show InChI InChI=1S/C25H22Cl2N4O2/c1-30-21-11-16-4-6-20(28-16)24(21)18-5-7-22(29-25(18)30)31-9-8-17(12-23(31)32)33-13-14-2-3-15(26)10-19(14)27/h2-3,5,7-10,12,16,20,28H,4,6,11,13H2,1H3
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 28 -43.1n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112704
PNG
(US8629158, 17)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(cc12)-n1ncc(OCc2ccc(F)cn2)cc1=O
Show InChI InChI=1S/C25H24FN5O2/c1-30-22-10-18(7-8-20(22)25-21-4-2-3-16(29-21)9-23(25)30)31-24(32)11-19(13-28-31)33-14-17-6-5-15(26)12-27-17/h5-8,10-13,16,21,29H,2-4,9,14H2,1H3
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 28 -43.1n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112726
PNG
(US8629158, 41)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C26H26N4O2/c1-29-22-14-18-8-5-9-21(27-18)25(22)20-10-11-23(28-26(20)29)30-13-12-19(15-24(30)31)32-16-17-6-3-2-4-7-17/h2-4,6-7,10-13,15,18,21,27H,5,8-9,14,16H2,1H3
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 30 -42.9n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112728
PNG
(US8629158, 43)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccc(F)cn2)cc1=O
Show InChI InChI=1S/C24H22FN5O2/c1-29-20-10-15-4-6-19(27-15)23(20)18-5-7-21(28-24(18)29)30-9-8-17(11-22(30)31)32-13-16-3-2-14(25)12-26-16/h2-3,5,7-9,11-12,15,19,27H,4,6,10,13H2,1H3
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 38 -42.4n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112695
PNG
(US8629158, 20 | US8629158, 21 | US8629158, 8)
Show SMILES O=c1cc(OCc2ccccc2)ccn1-c1ccc2c3C4CCC(Cc3[nH]c2c1)N4
Show InChI InChI=1S/C25H23N3O2/c29-24-14-19(30-15-16-4-2-1-3-5-16)10-11-28(24)18-7-8-20-22(13-18)27-23-12-17-6-9-21(26-17)25(20)23/h1-5,7-8,10-11,13-14,17,21,26-27H,6,9,12,15H2
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 39 -42.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112700
PNG
(US8629158, 13)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C26H23F3N4O/c1-32-21-13-18(6-7-19(21)25-20-4-2-3-17(31-20)12-22(25)32)33-10-9-15(11-24(33)34)16-5-8-23(30-14-16)26(27,28)29/h5-11,13-14,17,20,31H,2-4,12H2,1H3
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 46.3 -41.9n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112725
PNG
(US8629158, 40)
Show SMILES Cn1c2CC3CCCC(N3)c2c2ccc(nc12)-n1ccc(OCc2ccc(F)cn2)cc1=O
Show InChI InChI=1S/C25H24FN5O2/c1-30-21-11-16-3-2-4-20(28-16)24(21)19-7-8-22(29-25(19)30)31-10-9-18(12-23(31)32)33-14-17-6-5-15(26)13-27-17/h5-10,12-13,16,20,28H,2-4,11,14H2,1H3
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 49 -41.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112721
PNG
(US8629158, 35)
Show SMILES Cc1ccc(cn1)-c1ccn(-c2ccc3c4C5CCC(Cc4n(C)c3c2)N5)c(=O)c1
Show InChI InChI=1S/C25H24N4O/c1-15-3-4-17(14-26-15)16-9-10-29(24(30)11-16)19-6-7-20-22(13-19)28(2)23-12-18-5-8-21(27-18)25(20)23/h3-4,6-7,9-11,13-14,18,21,27H,5,8,12H2,1-2H3
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 59 -41.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112694
PNG
(US8629158, 7)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(cc12)-n1ccc(cc1=O)-c1cnc(nc1)C(F)(F)F |THB:10:9:8:6.5,1:2:8:6.5|
Show InChI InChI=1S/C24H20F3N5O/c1-31-19-10-16(3-4-17(19)22-18-5-2-15(30-18)9-20(22)31)32-7-6-13(8-21(32)33)14-11-28-23(29-12-14)24(25,26)27/h3-4,6-8,10-12,15,18,30H,2,5,9H2,1H3
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 68.1 -40.9n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112705
PNG
(US8629158, 18)
Show SMILES Cc1ccc(COc2cnn(-c3ccc4c5C6CCCC(Cc5n(C)c4c3)N6)c(=O)c2)cn1
Show InChI InChI=1S/C26H27N5O2/c1-16-6-7-17(13-27-16)15-33-20-12-25(32)31(28-14-20)19-8-9-21-23(11-19)30(2)24-10-18-4-3-5-22(29-18)26(21)24/h6-9,11-14,18,22,29H,3-5,10,15H2,1-2H3
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 73 -40.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112716
PNG
(US8629158, 29)
Show SMILES CC(=O)N1C2CCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccc(F)cn2)cc1=O |TLB:18:8:3:6.5,11:9:3:6.5|
Show InChI InChI=1S/C27H25FN4O3/c1-16(33)32-20-6-8-23(32)27-22-7-5-19(11-24(22)30(2)25(27)12-20)31-10-9-21(13-26(31)34)35-15-18-4-3-17(28)14-29-18/h3-5,7,9-11,13-14,20,23H,6,8,12,15H2,1-2H3
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 75 -40.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112717
PNG
(US8629158, 30)
Show SMILES CC(=O)N1C2CCC1c1c(C2)[nH]c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C27H25N3O3/c1-17(31)30-20-8-10-25(30)27-22-9-7-19(13-23(22)28-24(27)14-20)29-12-11-21(15-26(29)32)33-16-18-5-3-2-4-6-18/h2-7,9,11-13,15,20,25,28H,8,10,14,16H2,1H3
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 97 -40.0n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112731
PNG
(US8629158, 46)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)N1CCN(CCc2ccc(Cl)cc2)CC1=O
Show InChI InChI=1S/C25H28ClN5O/c1-29-21-14-18-6-8-20(27-18)24(21)19-7-9-22(28-25(19)29)31-13-12-30(15-23(31)32)11-10-16-2-4-17(26)5-3-16/h2-5,7,9,18,20,27H,6,8,10-15H2,1H3
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 99 -40.0n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112729
PNG
(US8629158, 44)
Show SMILES Cn1c2CC3CCC(N3)c2c2ccc(nc12)-n1ccc(cc1=O)-c1ccc(nc1)C(F)(F)F
Show InChI InChI=1S/C24H20F3N5O/c1-31-18-11-15-3-5-17(29-15)22(18)16-4-7-20(30-23(16)31)32-9-8-13(10-21(32)33)14-2-6-19(28-12-14)24(25,26)27/h2,4,6-10,12,15,17,29H,3,5,11H2,1H3
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 110 -39.7n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM112714
PNG
(US8629158, 27)
Show SMILES CC(=O)N1C2CCC1c1c(C2)n(C)c2cc(ccc12)-n1ccc(OCc2ccccc2)cc1=O
Show InChI InChI=1S/C28H27N3O3/c1-18(32)31-21-9-11-24(31)28-23-10-8-20(14-25(23)29(2)26(28)15-21)30-13-12-22(16-27(30)33)34-17-19-6-4-3-5-7-19/h3-8,10,12-14,16,21,24H,9,11,15,17H2,1-2H3
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 131 -39.3n/an/an/an/an/a7.425



Albany Molecular Research, Inc.

US Patent


Assay Description
Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...

US Patent US8629158 (2014)


BindingDB Entry DOI: 10.7270/Q24J0CS7
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%