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TargetCannabinoid receptor 2
LigandBDBM646493
Substrate/Competitorn/a
Meas. Tech.Inhibition of CB1, CB2 and A-Glucosidase by Kuwanon G and Albanin G Purified from Morus alba
IC50 28900±n/a nM
Citation Brownell, LAChoi, BCorneliusen, BHong, MHyun, EJia, QJiao, PKim, HKim, MKim, TLee, BLee, YNam, JYimam, MHwang, JOh, M Compositions and Methods for Managing Weight US Patent US20240024403 Publication Date 1/25/2024
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:39690.94
Organism:Homo sapiens (Human)
Description:P34972
Residue:360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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  Blast E-value cutoff:
BDBM646493
n/a
NameBDBM646493
Synonyms:US20240024403, Compound Kuwanon G
TypeSmall organic molecule
Emp. Form.C40H36O11
Mol. Mass.692.7072
SMILES[#6]\[#6](-[#6])=[#6]\[#6]-c1c(oc2c(-[#6]-3-[#6]=[#6](-[#6])-[#6]-[#6](-[#6]-3-[#6](=O)-c3ccc(-[#8])cc3-[#8])-c3ccc(-[#8])cc3-[#8])c(-[#8])cc(-[#8])c2c1=O)-c1ccc(-[#8])cc1-[#8] |t:11|
Structure
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