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TargetSimilar to alpha-tubulin isoform 1
LigandBDBM50472344
Substrate/Competitorn/a
Meas. Tech.ChEMBL_211318 (CHEMBL818978)
IC50 370±n/a nM
Citation Zhang, SXBastow, KFTachibana, YKuo, SCHamel, EMauger, ANarayanan, VLLee, KH Antitumor agents. 196. Substituted 2-thienyl-1,8-naphthyridin-4-ones: their synthesis, cytotoxicity, and inhibition of tubulin polymerization. J Med Chem42:4081-7 (1999) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Similar to alpha-tubulin isoform 1
Name:Similar to alpha-tubulin isoform 1
Synonyms:Similar to alpha-tubulin isoform 1
Type:PROTEIN
Mol. Mass.:10383.05
Organism:Bos taurus
Description:ChEMBL_104716
Residue:99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGK
HVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50472344
n/a
NameBDBM50472344
Synonyms:CHEMBL132896
TypeSmall organic molecule
Emp. Form.C17H12N2OS
Mol. Mass.292.355
SMILESCc1ccc2c(O)cc(nc2n1)-c1csc2ccccc12
Structure
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