| Reaction Details |
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 | Report a problem with these data |
| Target | Mas-related G-protein coupled receptor member X1 |
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| Ligand | BDBM50497458 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1436305 (CHEMBL3388386) |
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| EC50 | 1259±n/a nM |
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| Citation |  Hin, N; Alt, J; Zimmermann, SC; Delahanty, G; Ferraris, DV; Rojas, C; Li, F; Liu, Q; Dong, X; Slusher, BS; Tsukamoto, T Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors. Bioorg Med Chem22:5831-7 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mas-related G-protein coupled receptor member X1 |
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| Name: | Mas-related G-protein coupled receptor member X1 |
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| Synonyms: | MRGX1_MOUSE | Mas-related G-protein coupled receptor member C11 | Mas-related G-protein coupled receptor member X1 | Mrgc11 | Mrgprc11 | Mrgprx1 | Sensory neuron-specific G-protein coupled receptor 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36822.23 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_109490 |
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| Residue: | 322 |
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| Sequence: | MDPTISSHDTESTPLNETGHPNCTPILTLSFLVLITTLVGLAGNTIVLWLLGFRMRRKAI
SVYILNLALADSFFLCCHFIDSLLRIIDFYGLYAHKLSKDILGNAAIIPYISGLSILSAI
STERCLCVLWPIWYHCHRPRNMSAIICALIWVLSFLMGILDWFSGFLGETHHHLWKNVDF
IITAFLIFLFMLLSGSSLALLLRILCGPRRKPLSRLYVTIALTVMVYLICGLPLGLYLFL
LYWFGVHLHYPFCHIYQVTAVLSCVNSSANPIIYFLVGSFRQHRKHRSLKRVLKRALEDT
PEEDEYTDSHLHKTTEISESRY
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| BDBM50497458 |
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| n/a |
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| Name | BDBM50497458 |
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| Synonyms: | CHEMBL3343994 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H24N6O2 |
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| Mol. Mass. | 368.4329 |
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| SMILES | N[C@H](Cc1ccc(NC(N)=N)cc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r| |
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| Structure | 
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