| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 7 |
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| Ligand | BDBM50565197 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2091035 (CHEMBL4772298) |
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| Ki | 159±n/a nM |
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| Citation |  Jankowska, A; Sata?a, G; Ko?aczkowski, M; Bucki, A; G?uch-Lutwin, M; ?wierczek, A; Pociecha, K; Partyka, A; Jastrz?bska-Wi?sek, M; Lubelska, A; Latacz, G; Gawalska, A; Bojarski, AJ; Wyska, E; Ch?o?-Rzepa, G Novel anilide and benzylamide derivatives of arylpiperazinylalkanoic acids as 5-HT Eur J Med Chem201:0 (2020) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 7 |
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| Name: | 5-hydroxytryptamine receptor 7 |
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| Synonyms: | 5-HT-7 | 5-HT-X | 5-HT7 | 5-HT7L | 5-HT7S | 5-HT7b | 5HT7 | 5HT7R_HUMAN | HTR7 | Serotonin receptor 7 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 53573.08 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34969 |
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| Residue: | 479 |
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| Sequence: | MMDVNSSGRPDLYGHLRSFLLPEVGRGLPDLSPDGGADPVAGSWAPHLLSEVTASPAPTW
DAPPDNASGCGEQINYGRVEKVVIGSILTLITLLTIAGNCLVVISVCFVKKLRQPSNYLI
VSLALADLSVAVAVMPFVSVTDLIGGKWIFGHFFCNVFIAMDVMCCTASIMTLCVISIDR
YLGITRPLTYPVRQNGKCMAKMILSVWLLSASITLPPLFGWAQNVNDDKVCLISQDFGYT
IYSTAVAFYIPMSVMLFMYYQIYKAARKSAAKHKFPGFPRVEPDSVIALNGIVKLQKEVE
ECANLSRLLKHERKNISIFKREQKAATTLGIIVGAFTVCWLPFFLLSTARPFICGTSCSC
IPLWVERTFLWLGYANSLINPFIYAFFNRDLRTTYRSLLQCQYRNINRKLSAAGMHEALK
LAERPERPEFVLRACTRRVLLRPEKRPPVSVWVLQSPDHHNWLADKMLTTVEKKVMIHD
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| BDBM50565197 |
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| n/a |
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| Name | BDBM50565197 |
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| Synonyms: | CHEMBL4779965 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H38ClN3O3 |
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| Mol. Mass. | 476.051 |
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| SMILES | Cl.COc1ccccc1N1CCN(CCCCC(=O)Nc2cc(ccc2O)C(C)(C)C)CC1 |
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| Structure | 
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