Reaction Details |
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Target | Interleukin-17A |
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Ligand | BDBM50581143 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_2294275 |
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Kd | 660±n/a nM |
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Citation | Dimitrova, YN; Gutierrez, JA; Huard, K It's ok to be outnumbered - sub-stoichiometric modulation of homomeric protein complexes. RSC Med Chem14:22-46 (2023) [PubMed] |
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More Info.: | Get all data from this article, Assay Method |
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Interleukin-17A |
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Name: | Interleukin-17A |
Synonyms: | CTLA8 | Cytotoxic T-lymphocyte-associated antigen 8 | IL-17 | IL17 | IL17A | IL17_HUMAN | il-17a |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 17511.44 |
Organism: | Homo sapiens (Human) |
Description: | Q16552 |
Residue: | 155 |
Sequence: | MTPGKTSLVSLLLLLSLEAIVKAGITIPRNPGCPNSEDKNFPRTVMVNLNIHNRNTNTNP
KRSSDYYNRSTSPWNLHRNEDPERYPSVIWEAKCRHLGCINADGNVDYHMNSVPIQQEIL
VLRREPPHCPNSFRLEKILVSVGCTCVTPIVHHVA
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BDBM50581143 |
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n/a |
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Name | BDBM50581143 |
Synonyms: | CHEMBL5077648 |
Type | Small organic molecule |
Emp. Form. | C33H41FN6O4 |
Mol. Mass. | 604.7148 |
SMILES | CN(C)C(=O)CC1(CC(=O)NCCc2ccc(NC(=O)[C@H](Cc3ccccc3F)NC(=O)c3ccnn3C)cc2)CCCC1 |r| |
Structure |
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