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TargetInterleukin-17A
LigandBDBM50581143
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2294275
Kd 660±n/a nM
Citation Dimitrova, YNGutierrez, JAHuard, K It's ok to be outnumbered - sub-stoichiometric modulation of homomeric protein complexes. RSC Med Chem14:22-46 (2023) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Interleukin-17A
Name:Interleukin-17A
Synonyms:CTLA8 | Cytotoxic T-lymphocyte-associated antigen 8 | IL-17 | IL17 | IL17A | IL17_HUMAN | il-17a
Type:Enzyme Catalytic Domain
Mol. Mass.:17511.44
Organism:Homo sapiens (Human)
Description:Q16552
Residue:155
Sequence:
MTPGKTSLVSLLLLLSLEAIVKAGITIPRNPGCPNSEDKNFPRTVMVNLNIHNRNTNTNP
KRSSDYYNRSTSPWNLHRNEDPERYPSVIWEAKCRHLGCINADGNVDYHMNSVPIQQEIL
VLRREPPHCPNSFRLEKILVSVGCTCVTPIVHHVA
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50581143
n/a
NameBDBM50581143
Synonyms:CHEMBL5077648
TypeSmall organic molecule
Emp. Form.C33H41FN6O4
Mol. Mass.604.7148
SMILESCN(C)C(=O)CC1(CC(=O)NCCc2ccc(NC(=O)[C@H](Cc3ccccc3F)NC(=O)c3ccnn3C)cc2)CCCC1 |r|
Structure
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