| Reaction Details |
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 | Report a problem with these data |
| Target | Calcitonin gene-related peptide 1 |
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| Ligand | BDBM50246698 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_556924 (CHEMBL954950) |
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| IC50 | 1±n/a nM |
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| Citation |  Miranda, LP; Holder, JR; Shi, L; Bennett, B; Aral, J; Gegg, CV; Wright, M; Walker, K; Doellgast, G; Rogers, R; Li, H; Valladares, V; Salyers, K; Johnson, E; Wild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem51:7889-97 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Calcitonin gene-related peptide 1 |
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| Name: | Calcitonin gene-related peptide 1 |
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| Synonyms: | CALC1 | CALCA | CALCA_HUMAN | CGRP | Calcitonin gene-related peptide (CGRP alpha) | Calcitonin gene-related peptide 1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 13902.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P06881 |
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| Residue: | 128 |
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| Sequence: | MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQDYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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| BDBM50246698 |
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| n/a |
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| Name | BDBM50246698 |
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| Synonyms: | Ac-WVEHRLKGELSRKGGVV[hArg]KNFVPTDVGPFAF-NH2 | CHEMBL526728 |
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| Type | Small organic molecule |
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| Emp. Form. | C166H254N48O39 |
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| Mol. Mass. | 3546.0912 |
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| SMILES | n/a |
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| Structure | 
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