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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Mu-type opioid receptor | ||
| Ligand | BDBM50290889 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEBML_138751 | ||
| IC50 | >80000±n/a nM | ||
| Citation |  Liao, S; Lin, J; Shenderovich, MD; Han, Y; Hasohata, K; Davis, P; Qiu, W; Porreca, F; Yamamura, HI; Hruby, VJ The stereochemical requirements of the novel δ-opioid selective dipeptide antagonist TMT-Tic Bioorg Med Chem Lett7:3049-3052 (1997) Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Mu-type opioid receptor | |||
| Name: | Mu-type opioid receptor | ||
| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 11165.58 | ||
| Organism: | GUINEA PIG | ||
| Description: | P97266 | ||
| Residue: | 98 | ||
| Sequence: |
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| BDBM50290889 | |||
| n/a | |||
| Name | BDBM50290889 | ||
| Synonyms: | (S)-2-[(2R,3S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-butyryl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid; hydrochloride | CHEMBL545265 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C22H26N2O4 | ||
| Mol. Mass. | 382.4528 | ||
| SMILES | C[C@H]([C@@H](N)C(=O)N1Cc2ccccc2C[C@H]1C(O)=O)c1c(C)cc(O)cc1C |r| | ||
| Structure | 
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