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TargetSortase family protein
LigandBDBM50331605
Substrate/Competitorn/a
Meas. Tech.ChEMBL_687441 (CHEMBL1292117)
IC50 133000±n/a nM
Citation Lee, YJHan, YRPark, WNam, SHOh, KBLee, HS Synthetic analogs of indole-containing natural products as inhibitors of sortase A and isocitrate lyase. Bioorg Med Chem Lett20:6882-5 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sortase family protein
Name:Sortase family protein
Synonyms:Sortase | Sortase A (SrtA)
Type:Enzyme
Mol. Mass.:23546.15
Organism:Staphylococcus aureus
Description:n/a
Residue:206
Sequence:
MKKWTNRLMTIAGVVLILVAAYLFAKPHIDNYLHDKDKDEKIEQYDKNVKEQASKDKKQQ
AKPQIPKDKSKVAGYIEIPDADIKEPVYPGPATPEQLNRGVSFAEENESLDDQNISIAGH
TFIDRPNYQFTNLKAAKKGSMVYFKVGNETRKYKMTSIRDVKPTDVGVLDEQKGKDKQLT
LITCDDYNEKTGVWEKRKIFVATEVK
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  Blast E-value cutoff:
BDBM50331605
n/a
NameBDBM50331605
Synonyms:2-(2-methyl-1H-indol-3-yl)-2-oxoacetic acid | CHEMBL1288785
TypeSmall organic molecule
Emp. Form.C11H9NO3
Mol. Mass.203.1941
SMILESCc1[nH]c2ccccc2c1C(=O)C(O)=O
Structure
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