| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Serine/threonine-protein kinase 17B |
|---|
| Ligand | BDBM25919 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_774422 (CHEMBL1908639) |
|---|
| Kd | >10000±n/a nM |
|---|
| Citation |  Davis, MI; Hunt, JP; Herrgard, S; Ciceri, P; Wodicka, LM; Pallares, G; Hocker, M; Treiber, DK; Zarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol29:1046-51 (2011) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Serine/threonine-protein kinase 17B |
|---|
| Name: | Serine/threonine-protein kinase 17B |
|---|
| Synonyms: | DRAK2 | ST17B_HUMAN | STK17B | Serine/threonine-protein kinase 17B | Serine/threonine-protein kinase 17B (STK17B) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42332.49 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | O94768 |
|---|
| Residue: | 372 |
|---|
| Sequence: | MSRRRFDCRSISGLLTTTPQIPIKMENFNNFYILTSKELGRGKFAVVRQCISKSTGQEYA
AKFLKKRRRGQDCRAEILHEIAVLELAKSCPRVINLHEVYENTSEIILILEYAAGGEIFS
LCLPELAEMVSENDVIRLIKQILEGVYYLHQNNIVHLDLKPQNILLSSIYPLGDIKIVDF
GMSRKIGHACELREIMGTPEYLAPEILNYDPITTATDMWNIGIIAYMLLTHTSPFVGEDN
QETYLNISQVNVDYSEETFSSVSQLATDFIQSLLVKNPEKRPTAEICLSHSWLQQWDFEN
LFHPEETSSSSQTQDHSVRSSEDKTSKSSCNGTCGDREDKENIPEDSSMVSKRFRFDDSL
PNPHELVSDLLC
|
|
|
|---|
| BDBM25919 |
|---|
| n/a |
|---|
| Name | BDBM25919 |
|---|
| Synonyms: | BMS-345541 | BMS345541 | CHEMBL471496 | N-(2-aminoethyl)-3,12-dimethyl-2,5,8-triazatricyclo[7.4.0.0^{2,6}]trideca-1(13),3,5,7,9,11-hexaen-7-amine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C14H17N5 |
|---|
| Mol. Mass. | 255.3183 |
|---|
| SMILES | Cc1cnc2c(NCCN)nc3ccc(C)cc3n12 |
|---|
| Structure | 
|
|---|
Search and Browse
