| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50177894 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_302766 (CHEMBL838830) |
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| Ki | 2.1±n/a nM |
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| Citation |  Henriksen, G; Platzer, S; Hauser, A; Willoch, F; Berthele, A; Schwaiger, M; Wester, HJ 18F-labeled sufentanil for PET-imaging of mu-opioid receptors. Bioorg Med Chem Lett15:1773-7 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mor | OPIATE Mu | OPRM_MOUSE | Opioid receptors; mu and delta | Oprm | Oprm1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44431.62 |
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| Organism: | MOUSE |
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| Description: | OPIATE Mu OPRM1 MOUSE::P42866 |
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| Residue: | 398 |
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| Sequence: | MDSSAGPGNISDCSDPLAPASCSPAPGSWLNLSHVDGNQSDPCGPNRTGLGGSHSLCPQT
GSPSMVTAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATST
LPFQSVNYLMGTWPFGNILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRT
PRNAKIVNVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFA
FIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYV
IIKALITIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSTIEQ
QNSARIRQNTREHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM50177894 |
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| n/a |
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| Name | BDBM50177894 |
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| Synonyms: | 2-Fluoro-N-(1-phenethyl-piperidin-4-yl)-N-phenyl-propionamide | CHEMBL197479 | N-[1-[2-phenylethyl]-4-piperidinyl]-N-phenyl-2-[(+/-)-[18F]fluoropropanamide |
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| Type | Small organic molecule |
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| Emp. Form. | C22H27FN2O |
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| Mol. Mass. | 354.461 |
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| SMILES | CC(F)C(=O)N(C1CCN(CCc2ccccc2)CC1)c1ccccc1 |
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| Structure | 
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