| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Estrogen-related receptor gamma |
|---|
| Ligand | BDBM485070 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Binding Assay |
|---|
| IC50 | 53.0±n/a nM |
|---|
| Citation |  Hwang, SY; Cho, SJ; Kim, J; Chin, J; Hwang, H; Lee, I; Jeon, Y; Lee, J; Jeon, J; Kim, SW Aryl ethene derivative and pharmaceutical composition containing same as active ingredient US Patent US10934303 Publication Date 3/2/2021 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Estrogen-related receptor gamma |
|---|
| Name: | Estrogen-related receptor gamma |
|---|
| Synonyms: | ERR gamma-2 | ERR3 | ERR3_HUMAN | ERRG2 | ESRRG | Estrogen receptor-related protein 3 | Estrogen-Related Receptor, gamma | Estrogen-related receptor gamma | KIAA0832 | NR3B3 | Nuclear receptor subfamily 3 group B member 3 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 51305.00 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1501351 |
|---|
| Residue: | 458 |
|---|
| Sequence: | MDSVELCLPESFSLHYEEELLCRMSNKDRHIDSSCSSFIKTEPSSPASLTDSVNHHSPGG
SSDASGSYSSTMNGHQNGLDSPPLYPSAPILGGSGPVRKLYDDCSSTIVEDPQTKCEYML
NSMPKRLCLVCGDIASGYHYGVASCEACKAFFKRTIQGNIEYSCPATNECEITKRRRKSC
QACRFMKCLKVGMLKEGVRLDRVRGGRQKYKRRIDAENSPYLNPQLVQPAKKPYNKIVSH
LLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSL
LQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMK
LEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMT
LPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAKV
|
|
|
|---|
| BDBM485070 |
|---|
| n/a |
|---|
| Name | BDBM485070 |
|---|
| Synonyms: | US10934303, Cmpd No. 22q | US10934303, Example 68 | US11285226, Compound 22q |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C31H36N2O2 |
|---|
| Mol. Mass. | 468.6297 |
|---|
| SMILES | OCCC\C(=C(/c1ccc(O)cc1)c1ccc(cc1)N1CCN(CC1)C1CCC1)c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
