| Reaction Details |
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 | Report a problem with these data |
| Target | Bromodomain-containing protein 3 [51-123] |
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| Ligand | BDBM50370182 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Plate-Based Time-Resolved Fluorescence Energy Transfer (TR-FRET) Assays |
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| IC50 | 2275±n/a nM |
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| Citation |  Zhou, J; Brasier, AR; Tian, B; Liu, Z; Chen, H; Rytting, E Inhibitors of bromodomain-containing protein 4 (BRD4) US Patent US11117865 Publication Date 9/14/2021 |
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| More Info.: | Get all data from this article, Assay Method |
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| Bromodomain-containing protein 3 [51-123] |
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| Name: | Bromodomain-containing protein 3 [51-123] |
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| Synonyms: | BRD3 | BRD3_HUMAN | Bromodomain-containing protein 3 (BRD3)(BD1) | Bromodomain-containing protein 3 Bromo 1 domain(BRD3 BD1) | KIAA0043 | RING3L |
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| Type: | n/a |
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| Mol. Mass.: | 8887.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | BD1 (51-123 aa) of Q15059 |
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| Residue: | 73 |
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| Sequence: | WKHQFAWPFYQPVDAIKLNLPDYHKIIKNPMDMGTIKKRLENNYYWSASECMQDFNTMFT
NCYIYNKPTDDIV
|
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|
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| BDBM50370182 |
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| n/a |
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| Name | BDBM50370182 |
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| Synonyms: | CHEMBL4176038 | US11117865, Compound ZL0420 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H16N4O2 |
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| Mol. Mass. | 296.3238 |
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| SMILES | Cc1cc(\N=N\c2ccc3NC(=O)CCc3c2)c(N)cc1O |
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| Structure | 
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