| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 52 |
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| Ligand | BDBM622914 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Homogeneous Time-Resolved Fluorescence (HTRF) Assay |
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| EC50 | 3.00±n/a nM |
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| Citation |  Gerlach, K; Semple, G; Xiong, Y; Bertani, B; Ferrara, M; Fossati, G; Hobson, S; Lessel, UF; Runge, F; Mueller-Vieira, U; Wippich, J Substituted 3-phenoxyazetidin-1-yl-pyrazines US Patent US11780827 Publication Date 10/10/2023 |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 52 |
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| Name: | G-protein coupled receptor 52 |
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| Synonyms: | GPR52 | GPR52_HUMAN | Probable G-protein coupled receptor 52 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41366.15 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_108391 |
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| Residue: | 361 |
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| Sequence: | MNESRWTEWRILNMSSGIVNVSERHSCPLGFGHYSVVDVCIFETVVIVLLTFLIIAGNLT
VIFVFHCAPLLHHYTTSYFIQTMAYADLFVGVSCLVPTLSLLHYSTGVHESLTCQVFGYI
ISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIILIWIYSCLIFLPSFFGW
GKPGYHGDIFEWCATSWLTSAYFTGFIVCLLYAPAAFVVCFTYFHIFKICRQHTKEINDR
RARFPSHEVDSSRETGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSF
LTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCMCVKDQEAQEPKPRKRANSCS
I
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| BDBM622914 |
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| n/a |
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| Name | BDBM622914 |
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| Synonyms: | US11780827, Example 12 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H16F2N6O2 |
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| Mol. Mass. | 398.3661 |
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| SMILES | Cc1cc(NC(=O)c2nccnc2N2CC(C2)Oc2ccc(F)c(F)c2)cnn1 |
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| Structure | 
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