| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide FF receptor 1 |
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| Ligand | BDBM50500151 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1543522 (CHEMBL3750369) |
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| Ki | 1000±n/a nM |
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| Citation |  Keller, M; Weiss, S; Hutzler, C; Kuhn, KK; Mollereau, C; Dukorn, S; Schindler, L; Bernhardt, G; König, B; Buschauer, A N(?)-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([(3)H]UR-MK299) with Extended Residence Time. J Med Chem58:8834-49 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide FF receptor 1 |
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| Name: | Neuropeptide FF receptor 1 |
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| Synonyms: | G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47840.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1474637 |
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| Residue: | 430 |
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| Sequence: | MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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| BDBM50500151 |
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| n/a |
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| Name | BDBM50500151 |
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| Synonyms: | CHEMBL3746386 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H43F6N7O9 |
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| Mol. Mass. | 843.7692 |
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| SMILES | OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.CCC(=O)NCCNC(=O)\N=C(\N)NCCC[C@@H](NC(=O)C(c1ccccc1)c1ccccc1)C(=O)NCc1ccc(O)cc1 |r| |
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| Structure | 
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