| Reaction Details |
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 | Report a problem with these data |
| Target | Growth factor receptor-bound protein 2 |
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| Ligand | BDBM50066512 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_66901 (CHEMBL675383) |
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| IC50 | 1600±n/a nM |
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| Citation |  Furet, P; Gay, B; Caravatti, G; García-Echeverría, C; Rahuel, J; Schoepfer, J; Fretz, H Structure-based design and synthesis of high affinity tripeptide ligands of the Grb2-SH2 domain. J Med Chem41:3442-9 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Growth factor receptor-bound protein 2 |
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| Name: | Growth factor receptor-bound protein 2 |
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| Synonyms: | ASH | GRB2 | GRB2 adapter protein | GRB2_HUMAN | Grb2-SH2 | Growth factor receptor-bound protein 2 |
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| Type: | Protein |
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| Mol. Mass.: | 25205.04 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P62993 |
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| Residue: | 217 |
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| Sequence: | MEAIAKYDFKATADDELSFKRGDILKVLNEECDQNWYKAELNGKDGFIPKNYIEMKPHPW
FFGKIPRAKAEEMLSKQRHDGAFLIRESESAPGDFSLSVKFGNDVQHFKVLRDGAGKYFL
WVVKFNSLNELVDYHRSTSVSRNQQIFLRDIEQVPQQPTYVQALFDFDPQEDGELGFRRG
DFIHVMDNSDPNWWKGACHGQTGMFPRNYVTPVNRNV
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| BDBM50066512 |
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| n/a |
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| Name | BDBM50066512 |
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| Synonyms: | 2-(2-{2-Amino-3-[4-(diacetoxy-phosphoryloxy)-phenyl]-propionylamino}-hexanoylamino)-N-(2-ethyl-hexyl)-succinamic acid | CHEMBL113789 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H49N4O11P |
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| Mol. Mass. | 684.7147 |
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| SMILES | CCCCC(CC)CNC(=O)CC(NC(=O)C(CCCC)NC(=O)C(N)Cc1ccc(OP(=O)(OC(C)=O)OC(C)=O)cc1)C(O)=O |
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| Structure | 
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