| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 52 |
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| Ligand | BDBM50556709 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2056940 (CHEMBL4711941) |
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| IC50 | 2370±n/a nM |
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| Citation |  Wang, C; Zhang, YF; Guo, S; Zhao, Q; Zeng, Y; Xie, Z; Xie, X; Lu, B; Hu, Y GPR52 Antagonist Reduces Huntingtin Levels and Ameliorates Huntington's Disease-Related Phenotypes. J Med Chem64:941-957 (2021) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 52 |
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| Name: | G-protein coupled receptor 52 |
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| Synonyms: | GPR52 | GPR52_HUMAN | Probable G-protein coupled receptor 52 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41366.15 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_108391 |
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| Residue: | 361 |
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| Sequence: | MNESRWTEWRILNMSSGIVNVSERHSCPLGFGHYSVVDVCIFETVVIVLLTFLIIAGNLT
VIFVFHCAPLLHHYTTSYFIQTMAYADLFVGVSCLVPTLSLLHYSTGVHESLTCQVFGYI
ISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIILIWIYSCLIFLPSFFGW
GKPGYHGDIFEWCATSWLTSAYFTGFIVCLLYAPAAFVVCFTYFHIFKICRQHTKEINDR
RARFPSHEVDSSRETGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSF
LTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCMCVKDQEAQEPKPRKRANSCS
I
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| BDBM50556709 |
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| n/a |
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| Name | BDBM50556709 |
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| Synonyms: | CHEMBL4783011 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H15FO |
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| Mol. Mass. | 254.2988 |
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| SMILES | Fc1cccc(c1)C(=O)\C=C\CCc1ccccc1 |
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| Structure | 
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