Reaction Details |
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Target | Casein kinase II subunit alpha |
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Ligand | BDBM11323 |
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Substrate/Competitor | CK-2 Peptide Substrate |
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Meas. Tech. | Kinase Inhibition Assay |
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pH | 7.5±n/a |
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Temperature | 295.15±n/a K |
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Ki | 400±n/a nM |
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IC50 | 500±n/a nM |
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Citation | Sarno, S; de Moliner, E; Ruzzene, M; Pagano, MA; Battistutta, R; Bain, J; Fabbro, D; Schoepfer, J; Elliott, M; Furet, P; Meggio, F; Zanotti, G; Pinna, LA Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase CK2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin-7-yl]acetic acid (IQA). Biochem J374:639-46 (2003) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Casein kinase II subunit alpha |
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Name: | Casein kinase II subunit alpha |
Synonyms: | CK II | CK2 | CK2- alpha | CK2A1 | CSK21_HUMAN | CSNK2A1 | Casein kinase 2 | Casein kinase II (CK2) | Casein kinase II alpha/beta | Casein kinase II subunit alpha (CK2 alpha) | Casein kinase II subunit alpha (CK2A1) | Casein kinase II subunit alpha (CK2a I174A) | Casein kinase II subunit alpha (CK2a V66A) | Casein kinase II subunit alpha (CK2a dm V66I174AA) | Casein kinase II subunit alpha (CK2a) |
Type: | Enzyme |
Mol. Mass.: | 45151.12 |
Organism: | Homo sapiens (Human) |
Description: | P68400 |
Residue: | 391 |
Sequence: | MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINIT
NNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTD
FKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAE
FYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYD
QLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDF
LDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMGSSSMPGGSTPVSSANMMSGISSVPT
PSPLGPLAGSPVIAAANPLGMPVPAAAGAQQ
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BDBM11323 |
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CK-2 Peptide Substrate |
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Name: | CK-2 Peptide Substrate |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 1446.31 |
Organism: | n/a |
Description: | n/a |
Residue: | 12 |
Sequence: | |