| Reaction Details |
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 | Report a problem with these data |
| Target | Estrogen-related receptor gamma |
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| Ligand | BDBM20608 |
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| Substrate/Competitor | Biotinylated RIP140 peptide |
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| Meas. Tech. | ERRgamma FRET Assay |
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| pH | 7±n/a |
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| Temperature | 295.15±n/a K |
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| EC50 | 15±n/a nM |
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| Citation |  Zuercher, WJ; Gaillard, S; Orband-Miller, LA; Chao, EY; Shearer, BG; Jones, DG; Miller, AB; Collins, JL; McDonnell, DP; Willson, TM Identification and structure-activity relationship of phenolic acyl hydrazones as selective agonists for the estrogen-related orphan nuclear receptors ERRbeta and ERRgamma. J Med Chem48:3107-9 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Estrogen-related receptor gamma |
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| Name: | Estrogen-related receptor gamma |
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| Synonyms: | ERR gamma-2 | ERR3 | ERR3_HUMAN | ERRG2 | ESRRG | Estrogen receptor-related protein 3 | Estrogen-Related Receptor, gamma | Estrogen-related receptor gamma | KIAA0832 | NR3B3 | Nuclear receptor subfamily 3 group B member 3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 51305.00 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1501351 |
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| Residue: | 458 |
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| Sequence: | MDSVELCLPESFSLHYEEELLCRMSNKDRHIDSSCSSFIKTEPSSPASLTDSVNHHSPGG
SSDASGSYSSTMNGHQNGLDSPPLYPSAPILGGSGPVRKLYDDCSSTIVEDPQTKCEYML
NSMPKRLCLVCGDIASGYHYGVASCEACKAFFKRTIQGNIEYSCPATNECEITKRRRKSC
QACRFMKCLKVGMLKEGVRLDRVRGGRQKYKRRIDAENSPYLNPQLVQPAKKPYNKIVSH
LLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAKHIPGFSTLSLADQMSL
LQSAWMEILILGVVYRSLSFEDELVYADDYIMDEDQSKLAGLLDLNNAILQLVKKYKSMK
LEKEEFVTLKAIALANSDSMHIEDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMT
LPLLRQTSTKAVQHFYNIKLEGKVPMHKLFLEMLEAKV
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| BDBM20608 |
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| Biotinylated RIP140 peptide |
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| Name: | Biotinylated RIP140 peptide (aa 366-390) |
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| Synonyms: | NRIP1 | NRIP1_HUMAN | Nuclear factor RIP140, 366-390 | Receptor-interacting protein 140 derived peptide |
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| Type: | Peptide |
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| Mol. Mass.: | 2831.78 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P48552[366-390] |
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| Residue: | 25 |
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| Sequence: | LERNNIKQAANNSLLLHLLKSQTIP
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