| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 4 |
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| Ligand | BDBM261525 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | FLIPR Assay |
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| EC50 | 1658±n/a nM |
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| Citation |  Chelliah, M; Chu, HD; Cox, JM; Debenham, JS; Eagen, K; Lan, P; London, C; Plotkin, MA; Shah, U; Sinz, CJ; Sun, Z; Vaccaro, HM; Venkatraman, S Substituted spiropiperidinyl compounds useful as GPR120 agonists US Patent US9708270 Publication Date 7/18/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 4 |
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| Name: | Free fatty acid receptor 4 |
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| Synonyms: | FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42256.91 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1508994 |
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| Residue: | 377 |
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| Sequence: | MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVC
ALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTL
SGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVV
PQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQTSEHLLDA
RAVVTHSEITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITI
LLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGA
ILTDTSVKRNDLSIISG
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| BDBM261525 |
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| n/a |
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| Name | BDBM261525 |
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| Synonyms: | US9708270, 20 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H28FNO3 |
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| Mol. Mass. | 361.4503 |
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| SMILES | CCC(=O)c1ccc(F)c(c1)N1CCC2(CCC(CC(O)=O)CC2)CC1 |
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| Structure | 
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