Reaction Details |
| Report a problem with these data |
Target | DNA polymerase beta |
---|
Ligand | BDBM33391 |
---|
Substrate/Competitor | DNA template-primer |
---|
Meas. Tech. | DNA Polymerase Assay |
---|
pH | 7.5±n/a |
---|
Temperature | 310.15±n/a K |
---|
IC50 | >200000±n/a nM |
---|
Citation | Kuramochi, K; Fukudome, K; Kuriyama, I; Takeuchi, T; Sato, Y; Kamisuki, S; Tsubaki, K; Sugawara, F; Yoshida, H; Mizushina, Y Synthesis and structure-activity relationships of dehydroaltenusin derivatives as selective DNA polymerase alpha inhibitors. Bioorg Med Chem17:7227-38 (2009) [PubMed] Article |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
DNA polymerase beta |
---|
Name: | DNA polymerase beta |
Synonyms: | DNA Polymerase beta | DPOLB_RAT | Polb |
Type: | PROTEIN |
Mol. Mass.: | 38334.34 |
Organism: | Rattus norvegicus |
Description: | ChEMBL_1361926 |
Residue: | 335 |
Sequence: | MSKRKAPQETLNGGITDMLVELANFEKNVSQAIHKYNAYRKAASVIAKYPHKIKSGAEAK
KLPGVGTKIAEKIDEFLATGKLRKLEKIRQDDTSSSINFLTRVTGIGPSAARKLVDEGIK
TLEDLRKNEDKLNHHQRIGLKYFEDFEKRIPREEMLQMQDIVLNEVKKLDPEYIATVCGS
FRRGAESSGDMDVLLTHPNFTSESSKQPKLLHRVVEQLQKVRFITDTLSKGETKFMGVCQ
LPSENDENEYPHRRIDIRLIPKDQYYCGVLYFTGSDIFNKNMRAHALEKGFTINEYTIRP
LGVTGVAGEPLPVDSEQDIFDYIQWRYREPKDRSE
|
|
|
BDBM33391 |
---|
DNA template-primer |
---|
Name: | DNA template-primer |
Synonyms: | poly(dA)/oligo(dT)(12Â?1), A/T = 2/1 |
Type: | Duplex DNA |
Mol. Mass.: | 358.43 |
Organism: | n/a |
Description: | [3H]-dTTP as co-substrate. |
Residue: | 3 |
Sequence: | |