| Reaction Details |
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 | Report a problem with these data |
| Target | Dipeptidase 1 |
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| Ligand | BDBM36637 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dehydropeptidase I Assay |
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| pH | 7±0 |
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| Temperature | 310.15±0 K |
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| IC50 | >2.50e+5±n/a nM |
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| Citation |  Toney, JH; Fitzgerald, PM; Grover-Sharma, N; Olson, SH; May, WJ; Sundelof, JG; Vanderwall, DE; Cleary, KA; Grant, SK; Wu, JK; Kozarich, JW; Pompliano, DL; Hammond, GG Antibiotic sensitization using biphenyl tetrazoles as potent inhibitors of Bacteroides fragilis metallo-beta-lactamase. Chem Biol5:185-96 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Dipeptidase 1 |
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| Name: | Dipeptidase 1 |
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| Synonyms: | DPEP1 | DPEP1_HUMAN | Dehydropeptidase-I | Dehydropeptidase-I (DHP-1) | Dipeptidase 1 | MDP | Microsomal dipeptidase | RDP | Renal dipeptidase | hRDP |
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| Type: | Protein |
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| Mol. Mass.: | 45670.34 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P16444 |
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| Residue: | 411 |
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| Sequence: | MWSGWWLWPLVAVCTADFFRDEAERIMRDSPVIDGHNDLPWQLLDMFNNRLQDERANLTT
LAGTHTNIPKLRAGFVGGQFWSVYTPCDTQNKDAVRRTLEQMDVVHRMCRMYPETFLYVT
SSAGIRQAFREGKVASLIGVEGGHSIDSSLGVLRALYQLGMRYLTLTHSCNTPWADNWLV
DTGDSEPQSQGLSPFGQRVVKELNRLGVLIDLAHVSVATMKATLQLSRAPVIFSHSSAYS
VCASRRNVPDDVLRLVKQTDSLVMVNFYNNYISCTNKANLSQVADHLDHIKEVAGARAVG
FGGDFDGVPRVPEGLEDVSKYPDLIAELLRRNWTEAEVKGALADNLLRVFEAVEQASNLT
QAPEEEPIPLDQLGGSCRTHYGYSSGASSLHRHWGLLLASLAPLVLCLSLL
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| BDBM36637 |
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| n/a |
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| Name | BDBM36637 |
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| Synonyms: | L-809-558 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H15N7 |
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| Mol. Mass. | 353.38 |
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| SMILES | C(c1ccc(cc1)-c1ccccc1-c1nnn[nH]1)n1cnc2cccnc12 |
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| Structure | 
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