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TargetMu-type opioid receptor
LigandBDBM50010535
Substrate/Competitorn/a
Meas. Tech.ChEBML_146989
IC50 0.500000±n/a nM
Citation Yoshino HNakazawa TArakawa YKaneko TTsuchiya YMatsunaga MAraki SIkeda MYamatsu KTachibana S Synthesis and structure-activity relationships of dynorphin A-(1-8) amide analogues. J Med Chem 33:206-12 (1990) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50010535
n/a
NameBDBM50010535
Synonyms:2-{5-Guanidino-2-[(5-guanidino-2-{2-[2-(2-{2-[3-(4-hydroxy-phenyl)-2-methylamino-propionylamino]-acetylamino}-acetylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-pentanoyl)-methyl-amino]-pentanoylamino}-4-methyl-pentanoic acid amide | CHEMBL266035
TypeSmall organic molecule
Emp. Form.C48H77N15O9
Mol. Mass.1008.2201
SMILESCN[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)NCC(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N(C)[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(C)C)C(N)=O
Structure
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