| Reaction Details |
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 | Report a problem with these data |
| Target | Oxoeicosanoid receptor 1 |
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| Ligand | BDBM50275229 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1714532 (CHEMBL4124581) |
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| EC50 | >100000±n/a nM |
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| Citation |  Stepniewski, TM; Torrens-Fontanals, M; Rodríguez-Espigares, I; Giorgino, T; Primdahl, KG; Vik, A; Stenstrřm, Y; Selent, J; Hansen, TV Synthesis, molecular modelling studies and biological evaluation of new oxoeicosanoid receptor 1 agonists. Bioorg Med Chem26:3580-3587 (2018) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Oxoeicosanoid receptor 1 |
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| Name: | Oxoeicosanoid receptor 1 |
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| Synonyms: | 5-oxo-ETE G-protein coupled receptor | G-protein coupled receptor 170 | G-protein coupled receptor R527 | G-protein coupled receptor TG1019 | GPR170 | OXER1 | OXER1_HUMAN | Oxoeicosanoid receptor 1 | TG 1019 | TG1019 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 45833.20 |
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| Organism: | Homo sapiens (Human) |
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| Description: | TG 1019 0 HUMAN::Q8TDS5 |
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| Residue: | 423 |
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| Sequence: | MLCHRGGQLIVPIIPLCPEHSCRGRRLQNLLSGPWPKQPMELHNLSSPSPSLSSSVLPPS
FSPSPSSAPSAFTTVGGSSGGPCHPTSSSLVSAFLAPILALEFVLGLVGNSLALFIFCIH
TRPWTSNTVFLVSLVAADFLLISNLPLRVDYYLLHETWRFGAAACKVNLFMLSTNRTASV
VFLTAIALNRYLKVVQPHHVLSRASVGAAARVAGGLWVGILLLNGHLLLSTFSGPSCLSY
RVGTKPSASLRWHQALYLLEFFLPLALILFAIVSIGLTIRNRGLGGQAGPQRAMRVLAMV
VAVYTICFLPSIIFGMASMVAFWLSACRSLDLCTQLFHGSLAFTYLNSVLDPVLYCFSSP
NFLHQSRALLGLTRGRQGPVSDESSYQPSRQWRYREASRKAEAIGKLKVQGEVSLEKEGS
SQG
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| BDBM50275229 |
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| n/a |
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| Name | BDBM50275229 |
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| Synonyms: | CHEMBL4128214 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H32O3 |
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| Mol. Mass. | 356.4984 |
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| SMILES | CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/C=C/C(=O)CCC(=O)OC |
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| Structure | 
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