| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM82032 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_29452 (CHEMBL641037) |
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| Ki | 700±n/a nM |
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| Citation |  Peet, NP; Dickerson, GA; Abdallah, AH; Daly, JW; Ukena, D Benzo[1,2-c:5,4-c']dipyrazoles: non-xanthine adenosine antagonists. J Med Chem31:2034-9 (1988) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
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| Type: | Protein |
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| Mol. Mass.: | 36704.13 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | n/a |
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| Residue: | 326 |
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| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
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| BDBM82032 |
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| n/a |
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| Name | BDBM82032 |
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| Synonyms: | 1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Dipropylxanthine | CAS_169317 | CHEMBL157655 | CPX | NSC_169317 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H16N4O2 |
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| Mol. Mass. | 236.2703 |
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| SMILES | CCCn1c2nc[nH]c2c(=O)n(CCC)c1=O |
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| Structure | 
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