| Reaction Details |
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 | Report a problem with these data |
| Target | Vasopressin V2 receptor |
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| Ligand | BDBM50452524 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_214849 |
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| Ki | 3.6±n/a nM |
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| Citation |  Moore, ML; Albrightson, C; Brickson, B; Bryan, HG; Caldwell, N; Callahan, JF; Foster, J; Kinter, LB; Newlander, KA; Schmidt, DB Dicarbavasopressin antagonist analogues exhibit reduced in vivo agonist activity. J Med Chem31:1487-9 (1988) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Vasopressin V2 receptor |
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| Name: | Vasopressin V2 receptor |
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| Synonyms: | AVPR2 | V2R_PIG |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40556.17 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_214870 |
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| Residue: | 370 |
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| Sequence: | MLRATTSAVPRALSWPAAPGNGSEREPLDDRDPLLARVELALLSTVFVAVALSNGLVLGA
LVRRGRRGRWAPMHVFIGHLCLADLAVALFQVLPQLAWDATYRFRGPDALCRAVKYLQMV
GMYASSYMILAMTLDRHRAICRPMLAYRHGGGARWNRPVLVAWAFSLLLSLPQLFIFAQR
DVGDGSGVLDCWASFAEPWGLRAYVTWIALMVFVAPALGIAACQVLIFREIHTSLVPGPA
ERAGGHRGGRRAGSPREGARVSAAMAKTARMTLVIVAVYVLCWAPFFLVQLWSVWDPKAP
REGPPFVLLMLLASLNSCTNPWIYASFSSSISSELRSLLCCPRRRTPPSLRPQEESCATA
SSFSARDTSS
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| BDBM50452524 |
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| n/a |
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| Name | BDBM50452524 |
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| Synonyms: | CHEMBL2372291 |
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| Type | Small organic molecule |
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| Emp. Form. | C51H74N12O10S2 |
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| Mol. Mass. | 1079.338 |
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| SMILES | [#6]-[#6]-[#8]-c1ccc(-[#6]-[#6@H]-2-[#7]-[#6](=O)-[#6]C3([#6]-[#6]-[#6]-[#6]-[#6]3)[#16]-[#16]-[#6]-[#6](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-c3ccccc3)-[#7]-[#6]-2=O)-[#6](-[#6])-[#6])-[#6](=O)-[#7]-2-[#6]-[#6]-[#6]-[#6@@H]-2-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](-[#7])=O)cc1 |
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| Structure | 
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