| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Mu-type opioid receptor |
|---|
| Ligand | BDBM50140906 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_221917 (CHEMBL842482) |
|---|
| IC50 | 21±n/a nM |
|---|
| Citation |  Yamazaki, T; Ro, S; Goodman, M; Chung, NN; Schiller, PW A topochemical approach to explain morphiceptin bioactivity. J Med Chem36:708-19 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Mu-type opioid receptor |
|---|
| Name: | Mu-type opioid receptor |
|---|
| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 11165.58 |
|---|
| Organism: | GUINEA PIG |
|---|
| Description: | P97266 |
|---|
| Residue: | 98 |
|---|
| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
|
|
|---|
| BDBM50140906 |
|---|
| n/a |
|---|
| Name | BDBM50140906 |
|---|
| Synonyms: | 1-[2-[1-[2-amino-3-(4-hydroxyphenyl)-(2S)-propanoyl]-(5S)-dihydro-1H-5-pyrrolyl(methyl)carboxamido]-3-phenyl-(2S)-propanoyl]-(5R)-dihydro-1H-5-pyrrolecarboxamide | CHEMBL283287 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C29H37N5O5 |
|---|
| Mol. Mass. | 535.6346 |
|---|
| SMILES | CN([C@@H](Cc1ccccc1)C(=O)N1CCC[C@@H]1C(N)=O)C(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
