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TargetChymotrypsinogen A
LigandBDBM26139
Substrate/Competitorn/a
Meas. Tech.ChEMBL_34119 (CHEMBL649747)
IC50 5000±n/a nM
Citation Weston, GSBlázquez, JBaquero, FShoichet, BK Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase. J Med Chem41:4577-86 (1998) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Chymotrypsinogen A
Name:Chymotrypsinogen A
Synonyms:Alpha-chymotrypsin | CTRA_BOVIN | Chymotrypsin A | Chymotrypsin A chain A | Chymotrypsin A chain B | Chymotrypsin A chain C | Chymotrypsinogen A | alpha-Chymotrypsin (α-Chymotrypsin)
Type:Serine protease
Mol. Mass.:25670.88
Organism:Bos taurus (bovine)
Description:n/a
Residue:245
Sequence:
CGVPAIQPVLSGLSRIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGV
TTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSA
VCLPSASDDFAAGTTCVTTGWGLTRYTNANTPDRLQQASLPLLSNTNCKKYWGTKIKDAM
ICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQ
TLAAN
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BDBM26139
n/a
NameBDBM26139
Synonyms:1-benzothiophen-2-ylboranediol | 1-benzothiophen-2-ylboronic acid, 18 | CHEMBL34964 | Phenylboronic acid, 11
Typen/a
Emp. Form.C8H7BO2S
Mol. Mass.178.016
SMILESOB(O)c1cc2ccccc2s1
Structure
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