| Reaction Details |
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 | Report a problem with these data |
| Target | Serine protease 1 |
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| Ligand | BDBM50070790 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_212738 |
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| Ki | 233000±n/a nM |
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| Citation |  Naylor-Olsen, AM; Ponticello, GS; Lewis, SD; Mulichak, AM; Chen, Z; Habecker, CN; Phillips, BT; Sanders, WM; Tucker, TJ; Shafer, JA; Vacca, JP Identification and SAR for a selective, nonpeptidyl thrombin inhibitor. Bioorg Med Chem Lett8:1697-702 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Serine protease 1 |
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| Name: | Serine protease 1 |
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| Synonyms: | Alpha-trypsin chain 1 | Alpha-trypsin chain 2 | Beta-trypsin | Cationic trypsinogen | PRSS1 | Serine protease 1 | TRP1 | TRY1 | TRY1_HUMAN | TRYP1 | Thrombin & trypsin | Trypsin | Trypsin I | Trypsin-1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 26557.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P07477 |
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| Residue: | 247 |
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| Sequence: | MNPLLILTFVAAALAAPFDDDDKIVGGYNCEENSVPYQVSLNSGYHFCGGSLINEQWVVS
AGHCYKSRIQVRLGEHNIEVLEGNEQFINAAKIIRHPQYDRKTLNNDIMLIKLSSRAVIN
ARVSTISLPTAPPATGTKCLISGWGNTASSGADYPDELQCLDAPVLSQAKCEASYPGKIT
SNMFCVGFLEGGKDSCQGDSGGPVVCNGQLQGVVSWGDGCAQKNKPGVYTKVYNYVKWIK
NTIAANS
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| BDBM50070790 |
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| n/a |
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| Name | BDBM50070790 |
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| Synonyms: | (4-Benzyloxy-benzyl)-pyridin-4-yl-amine | CHEMBL47751 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H18N2O |
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| Mol. Mass. | 290.359 |
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| SMILES | C(Nc1ccncc1)c1ccc(OCc2ccccc2)cc1 |
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| Structure | 
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