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TargetHistamine H3 receptor
LigandBDBM22915
Substrate/Competitorn/a
Meas. Tech.ChEBML_86751
Ki 2.9±n/a nM
Citation Stark HSippl WLigneau XArrang JMGanellin CRSchwartz JCSchunack W Different antagonist binding properties of human and rat histamine H3 receptors. Bioorg Med Chem Lett 11:951-4 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Histamine H3 receptor
Name:Histamine H3 receptor
Synonyms:HH3R
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:48607.98
Organism:Rattus norvegicus (rat)
Description:n/a
Residue:445
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFV
ADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCAS
SVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGG
SSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAG
PEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRYGVGEAGPGVEAGEAALGGGSGGGAA
ASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSL
AIIVSIFGLCWAPYTLLMIIRAACHGRCIPDYWYETSFWLLWANSAVNPVLYPLCHYSFR
RAFTKLLCPQKLKVQPHGSLEQCWK
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  Blast E-value cutoff:
BDBM22915
n/a
NameBDBM22915
Synonyms:3-(1H-imidazol-4-yl)propylphenylmethyl ether | 5-[3-(benzyloxy)propyl]-1H-imidazole | CHEMBL61618 | PROXYFAN | Proxyfan
TypeSmall organic molecule
Emp. Form.C13H16N2O
Mol. Mass.216.2789
SMILESC(COCc1ccccc1)Cc1cnc[nH]1
Structure
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