| Reaction Details |
|---|
 | Report a problem with these data |
| Target | D(3) dopamine receptor |
|---|
| Ligand | BDBM50580522 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_2148518 (CHEMBL5032916) |
|---|
| Ki | 364±n/a nM |
|---|
| Citation |  Hagenow, S; Affini, A; Pioli, EY; Hinz, S; Zhao, Y; Porras, G; Namasivayam, V; Müller, CE; Lin, JS; Bezard, E; Stark, H Adenosine A J Med Chem64:8246-8262 (2021) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| D(3) dopamine receptor |
|---|
| Name: | D(3) dopamine receptor |
|---|
| Synonyms: | DRD3 | DRD3_HUMAN | Dopamine D3 receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 44213.40 |
|---|
| Organism: | Homo sapiens |
|---|
| Description: | ChEMBL_105671 |
|---|
| Residue: | 400 |
|---|
| Sequence: | MASLSQLSGHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
|
|
|
|---|
| BDBM50580522 |
|---|
| n/a |
|---|
| Name | BDBM50580522 |
|---|
| Synonyms: | CHEMBL5082650 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H26N4O2 |
|---|
| Mol. Mass. | 414.4995 |
|---|
| SMILES | Nc1nc2-c3cc(OCCCN4CCCCC4)ccc3C(=O)c2c(n1)-c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
