| Reaction Details |
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 | Report a problem with these data |
| Target | Peroxisome proliferator-activated receptor gamma |
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| Ligand | BDBM50208865 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_455158 (CHEMBL887188) |
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| EC50 | 200±n/a nM |
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| Citation |  Sauerberg, P; Mogensen, JP; Jeppesen, L; Bury, PS; Fleckner, J; Olsen, GS; Jeppesen, CB; Wulff, EM; Pihera, P; Havranek, M; Polivka, Z; Pettersson, I Design of potent PPARalpha agonists. Bioorg Med Chem Lett17:3198-202 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Peroxisome proliferator-activated receptor gamma |
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| Name: | Peroxisome proliferator-activated receptor gamma |
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| Synonyms: | NR1C3 | Nuclear receptor subfamily 1 group C member 3 | PPAR-gamma | PPARG | PPARG_HUMAN | Peroxisome proliferator-activated receptor | Peroxisome proliferator-activated receptor gamma (PPAR gamma) | Peroxisome proliferator-activated receptor gamma (PPARG) | Peroxisome proliferator-activated receptor gamma (PPARĪ³) | Peroxisome proliferator-activated receptor gamma/Nuclear receptor corepressor 2 | peroxisome proliferator-activated receptor gamma isoform 2 |
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| Type: | Nuclear Receptor |
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| Mol. Mass.: | 57613.46 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P37231 |
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| Residue: | 505 |
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| Sequence: | MGETLGDSPIDPESDSFTDTLSANISQEMTMVDTEMPFWPTNFGISSVDLSVMEDHSHSF
DIKPFTTVDFSSISTPHYEDIPFTRTDPVVADYKYDLKLQEYQSAIKVEPASPPYYSEKT
QLYNKPHEEPSNSLMAIECRVCGDKASGFHYGVHACEGCKGFFRRTIRLKLIYDRCDLNC
RIHKKSRNKCQYCRFQKCLAVGMSHNAIRFGRMPQAEKEKLLAEISSDIDQLNPESADLR
ALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQE
QSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLAS
LMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVII
LSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQL
LQVIKKTETDMSLHPLLQEIYKDLY
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| BDBM50208865 |
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| n/a |
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| Name | BDBM50208865 |
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| Synonyms: | (S)-3-(4-(3,5-diethoxycinnamyloxy)phenyl)-2-ethoxypropanoic acid | CHEMBL248113 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H30O6 |
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| Mol. Mass. | 414.4914 |
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| SMILES | CCO[C@@H](Cc1ccc(OC\C=C\c2cc(OCC)cc(OCC)c2)cc1)C(O)=O |
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| Structure | 
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