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TargetCannabinoid receptor 2
LigandBDBM50219073
Substrate/Competitorn/a
Meas. Tech.ChEMBL_445330
Ki 1.7±n/a nM
Citation Papahatjis DPNahmias VRNikas SPAndreou TAlapafuja SOTsotinis AGuo JFan PMakriyannis A C1'-cycloalkyl side chain pharmacophore in tetrahydrocannabinols. J Med Chem 50:4048-60 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CNR2 | Cannabinoid CB2 receptor | Cannabinoid receptor | mCB2
Type:Enzyme Catalytic Domain
Mol. Mass.:38220.43
Organism:MOUSE
Description:P47936
Residue:347
Sequence:
MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50219073
n/a
NameBDBM50219073
Synonyms:(6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclopropyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol | CHEMBL231465
TypeSmall organic molecule
Emp. Form.C25H34O2
Mol. Mass.366.5363
SMILESCCCC\C=C/C1(CC1)c1cc(O)c2[C@@H]3CC(C)=CC[C@H]3C(C)(C)Oc2c1 |c:18|
Structure
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