| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50219073 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_445330 (CHEMBL894470) |
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| Ki | 1.7±n/a nM |
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| Citation |  Papahatjis, DP; Nahmias, VR; Nikas, SP; Andreou, T; Alapafuja, SO; Tsotinis, A; Guo, J; Fan, P; Makriyannis, A C1'-cycloalkyl side chain pharmacophore in tetrahydrocannabinols. J Med Chem50:4048-60 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38220.43 |
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| Organism: | MOUSE |
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| Description: | P47936 |
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| Residue: | 347 |
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| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
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| BDBM50219073 |
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| n/a |
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| Name | BDBM50219073 |
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| Synonyms: | (6aR-trans)-3-[1-[(1Z)-1-hexenyl]cyclopropyl]-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-1-ol | CHEMBL231465 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H34O2 |
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| Mol. Mass. | 366.5363 |
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| SMILES | CCCC\C=C/C1(CC1)c1cc(O)c2[C@@H]3CC(C)=CC[C@H]3C(C)(C)Oc2c1 |c:18| |
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| Structure | 
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