| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50251029 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_529941 (CHEMBL975012) |
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| Ki | 78±n/a nM |
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| Citation |  Sipos, A; Kiss, B; Schmidt, E; Greiner, I; Berényi, S Synthesis and neuropharmacological evaluation of 2-aryl- and alkylapomorphines. Bioorg Med Chem16:3773-9 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3_RAT | Dopamine D3 receptor | Drd3 |
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| Type: | Protein |
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| Mol. Mass.: | 49540.58 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | P19020 |
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| Residue: | 446 |
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| Sequence: | MAPLSQISTHLNSTCGAENSTGVNRARPHAYYALSYCALILAIIFGNGLVCAAVLRERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPSI
CSISNPDFVIYSSVVSFYVPFGVTVLVYARIYIVLRQRQRKRILTRQNSQCISIRPGFPQ
QSSCLRLHPIRQFSIRARFLSDATGQMEHIEDKQYPQKCQDPLLSHLQPPSPGQTHGGLK
RYYSICQDTALRHPSLEGGAGMSPVERTRNSLSPTMAPKLSLEVRKLSNGRLSTSLRLGP
LQPRGVPLREKKATQMVVIVLGAFIVCWLPFFLTHVLNTHCQACHVSPELYRATTWLGYV
NSALNPVIYTTFNVEFRKAFLKILSC
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| BDBM50251029 |
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| n/a |
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| Name | BDBM50251029 |
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| Synonyms: | (R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine dihydrochloride | CHEMBL458587 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H26N2O2 |
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| Mol. Mass. | 386.4861 |
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| SMILES | CN(C)c1ccc(cc1)-c1cc2CCN(C)[C@@H]3Cc4ccc(O)c(O)c4-c(c1)c23 |r| |
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| Structure | 
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