| Reaction Details |
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 | Report a problem with these data |
| Target | Protein ADM2 |
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| Ligand | BDBM50246709 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_556927 (CHEMBL954953) |
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| IC50 | 418±n/a nM |
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| Citation |  Miranda, LP; Holder, JR; Shi, L; Bennett, B; Aral, J; Gegg, CV; Wright, M; Walker, K; Doellgast, G; Rogers, R; Li, H; Valladares, V; Salyers, K; Johnson, E; Wild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem51:7889-97 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein ADM2 |
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| Name: | Protein ADM2 |
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| Synonyms: | ADM2 | ADM2_HUMAN | AM2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 15883.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_556927 |
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| Residue: | 148 |
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| Sequence: | MARIPTAALGCISLLCLQLPGSLSRSLGGDPRPVKPREPPARSPSSSLQPRHPAPRPVVW
KLHRALQAQRGAGLAPVMGQPLRDGGRQHSGPRRHSGPRRTQAQLLRVGCVLGTCQVQNL
SHRLWQLMGPAGRQDSAPVDPSSPHSYG
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| BDBM50246709 |
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| n/a |
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| Name | BDBM50246709 |
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| Synonyms: | Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[2-Nal]AF-NH2 | CHEMBL509603 |
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| Type | Small organic molecule |
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| Emp. Form. | C164H248N44O41 |
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| Mol. Mass. | 3491.9941 |
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| SMILES | n/a |
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| Structure | 
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