| Reaction Details |
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 | Report a problem with these data |
| Target | Chymotrypsin-like elastase family member 2A |
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| Ligand | BDBM50281094 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_194721 |
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| IC50 | >200000±n/a nM |
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| Citation |  Adonias, M; Anayaba, J; Cámara, J; Canet, E; Gateau-Olesker, A; Gero, SD; Grande, M; Hernando, JI Enantioselective synthesis and antielastase activity of 1,3,4-trisubstituted and 3,4-disubstituted β-lactam antibiotics Bioorg Med Chem Lett3:2547-2552 (1993) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Chymotrypsin-like elastase family member 2A |
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| Name: | Chymotrypsin-like elastase family member 2A |
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| Synonyms: | CEL2A_RAT | Cela2a | Ela2 | Ela2a | Elastase 2A | Elastase-2 | Elastase-2A |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28894.94 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_194721 |
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| Residue: | 271 |
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| Sequence: | MIRTLLLSALVAGALSCGYPTYEVQHDVSRVVGGQEASPNSWPWQVSLQYLSSGKWHHTC
GGSLVANNWVLTAAHCISNSRTYRVLLGRHSLSTSESGSLAVQVSKLVVHEKWNAQKLSN
GNDIALVKLASPVALTSKIQTACLPPAGTILPNNYPCYVTGWGRLQTNGATPDVLQQGRL
LVVDYATCSSASWWGSSVKTNMVCAGGDGVTSSCNGDSGGPLNCQASNGQWQVHGIVSFG
STLGCNYPRKPSVFTRVSNYIDWINSVIAKN
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| BDBM50281094 |
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| n/a |
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| Name | BDBM50281094 |
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| Synonyms: | (3R,4R)-3-Butyl-1-[(R)-[1,3]dithian-2-yl-(2,2,2',2'-tetramethyl-[4,4']bi[[1,3]dioxolanyl]-5-yl)-methyl]-4-((E)-1-methyl-2-phenyl-vinyl)-azetidin-2-one | CHEMBL82333 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H45NO5S2 |
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| Mol. Mass. | 575.823 |
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| SMILES | CCCC[C@@H]1[C@@H](N([C@H](C2OC(C)(C)OC2C2COC(C)(C)O2)C2SCCCS2)C1=O)C(\C)=C\c1ccccc1 |
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| Structure | 
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