| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM50290032 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_58462 |
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| Ki | >1600±n/a nM |
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| Citation |  Haworth, KE; Harrison, T; Kulagowski, JJ; Leeson, PD; Owens, AP; Ridgill, MP; Teall, MR; Fielding, M; Chapman, K; Emms, F; Marwood, R; Patel, S; Moss, KL 4-Heterocyclyl tetrahydropyridines as selective ligands for the human dopamine D4 receptor Bioorg Med Chem Lett7:2211-2216 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | D(2) dopamine receptor | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2 | DRD2_HUMAN | Dopamine D2 receptor | Dopamine D2 receptor (D2) | Dopamine D2 receptor (D2R) | Dopamine D2A | Dopamine2-like | d2 |
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| Type: | Cell-surface receptors |
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| Mol. Mass.: | 50647.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P14416 |
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| Residue: | 443 |
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| Sequence: | MDPLNLSWYDDDLERQNWSRPFNGSDGKADRPHYNYYATLLTLLIAVIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMISIVWVLSFTISCPLLFGLNNADQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRAHLRAPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKDHPKIAKIFEIQTMPNGKTRTSLKTMSR
RKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSA
VNPIIYTTFNIEFRKAFLKILHC
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| BDBM50290032 |
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| n/a |
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| Name | BDBM50290032 |
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| Synonyms: | 2-[1-(4-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole | CHEMBL306265 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H17ClN2S |
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| Mol. Mass. | 340.87 |
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| SMILES | Clc1ccc(CN2CCC(=CC2)c2nc3ccccc3s2)cc1 |c:9| |
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| Structure | 
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